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Found 3 Enz. Inhib. hit(s) with Target = 'Sphingosine 1-phosphate receptor 5' and Ligand = 'BDBM321316'
TargetSphingosine 1-phosphate receptor 5(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM321316(US10179791, Compound 140 | US10807991, Compound 14...)
Affinity DataEC50:  3.16nMAssay Description:The CHO-human-S1P5-Aeqorin assay was bought from Euroscreen, Brussels (Euroscreen, Technical dossier, Human Lysophospholid S1P5 (Edg8) receptor, DNA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 5(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM321316(US10179791, Compound 140 | US10807991, Compound 14...)
Affinity DataEC50:  3.16nMAssay Description:The CHO-human-S1P5-Aeqorin assay was bought from Euroscreen, Brussels (Euroscreen, Technical dossier, Human Lysophospholid S1P5 (Edg8) receptor, DNA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 5(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM321316(US10179791, Compound 140 | US10807991, Compound 14...)
Affinity DataEC50:  2.5nMAssay Description:Agonist activity at human S1P5 receptor expressed in CHO cells assessed as increase in calcium flux by aequorin-derived luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed