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Found 3 Enz. Inhib. hit(s) with Target = 'Transmembrane domain-containing protein TMIGD3' and Ligand = 'BDBM50500484'
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500484(CHEMBL3745868)
Affinity DataKi:  33.9nMAssay Description:Displacement of CA200645 from human adenosine A3 receptor expressed in CHO CRE-SPAP cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500484(CHEMBL3745868)
Affinity DataKi:  34nMAssay Description:Displacement of CA200645 from human adenosine A3 receptor expressed in CHO CRE-SPAP cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500484(CHEMBL3745868)
Affinity DataKd:  741nMAssay Description:Competitive antagonist activity at YFP linked human adenosine A3 receptor expressed in CHO CRE-SPAP cells assessed as inhibition of NECA-induced rece...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed