Found 29 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase ABL1' and Ligand = 'BDBM50237710'
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 1.20nMAssay Description:Inhibition of recombinant human N-terminal His-tagged Abl (2 to 1130 residues) expressed in baculovirus expression system using FAM-labelled P2 pepti...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 5.60nMAssay Description:Inhibition of human ABL1 assessed as residual activity using EAIYAAPFAKKK as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 19nMAssay Description:Inhibition of ABL1 (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 28nMAssay Description:Inhibition of kinobead binding to ABL in human K562 cells incubated for 30 mins by iTRAQ reagent-based mass spectrometric methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 30nMAssay Description:Inhibition of full-length N-terminal His-tagged human c-Abl kinase (2 to 1130 residues) expressed in baculovirus expression system using Tk-substrate...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 30nMAssay Description:Inhibition of Abl (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 38nMAssay Description:Inhibition of wild type AblMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 44nMAssay Description:Inhibition of human recombinant wild type ABL1 expressed in insect cells after 30 mins by FRET assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 120nMAssay Description:In vitro kinase assay using Abl, Abl T315I or Src kinase.More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 9.17E+3nMAssay Description:Inhibition of ABL1 T315I mutant (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataKd: 10nMAssay Description:Binding constant for ABL1-nonphosphorylated kinase domainMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataKd: 21nMAssay Description:Binding constant for ABL1(Q252H)-phosphorylated kinase domainMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataKd: 36nMAssay Description:Binding constant for ABL1(E255K)-phosphorylated kinase domainMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataKd: 21nMAssay Description:Binding constant for ABL1(H396P)-phosphorylated kinase domainMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataKd: 14nMAssay Description:Binding constant for ABL1(F317L)-phosphorylated kinase domainMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataKd: 3.60nMAssay Description:Binding affinity to human ABL1More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataKd: 13nMAssay Description:Binding constant for ABL1(Y253F)-phosphorylated kinase domainMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataKd: 4.90nMAssay Description:Binding affinity to ABL1 (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ABL1(T315I)-phosphorylated kinase domainMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataKd: 56nMAssay Description:Binding constant for ABL1(F317I)-phosphorylated kinase domainMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataKd: 10nMAssay Description:Binding constant for ABL1(Q252H)-nonphosphorylated kinase domainMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataKd: 12nMAssay Description:Binding constant for ABL1(F317L)-nonphosphorylated kinase domainMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataKd: 18nMAssay Description:Binding constant for ABL1(F317I)-nonphosphorylated kinase domainMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataKd: 4.90nMAssay Description:Binding constant for ABL1(H396P)-nonphosphorylated kinase domainMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataKd: 13nMAssay Description:Binding constant for ABL1-phosphorylated kinase domainMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataKd: 15nMAssay Description:Binding constant for ABL1(M351T)-phosphorylated kinase domainMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataKd: 660nMAssay Description:Binding constant for ABL1(T315I)-nonphosphorylated kinase domainMore data for this Ligand-Target Pair