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Found 2 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase BTK' and Ligand = 'BDBM465744'
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM465744(2-{3-[2-amino-6-(pyridin-4-yl)-7H- pyrrolo[2,3-d]p...)
Affinity DataIC50:  0.140nMAssay Description:Inhibition of human BTK-A using phosphorylated substrate in presence of ATP by microplate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM465744(2-{3-[2-amino-6-(pyridin-4-yl)-7H- pyrrolo[2,3-d]p...)
Affinity DataIC50: <10nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trade mark) MSA (commercially available kit manufactured by Carna Biosciences, In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent