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Found 3 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase JAK1' and Ligand = 'BDBM26198'
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
University Of Luxembourg

LigandPNGBDBM26198(4-tert-butyl-15-fluoro-3,5,10-triazatetracyclo[11....)
Affinity DataIC50:  5.20nMpH: 7.5 T: 2°CAssay Description:Enzyme assay affinity-purified GST fusions of the active kinase domains (GST-Jak1(866-1154), GST-Jak2(808-1132), GST-Jak3(811-1124) and GST-Tyk2(888-...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK1(Mus musculus)
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM26198(4-tert-butyl-15-fluoro-3,5,10-triazatetracyclo[11....)
Affinity DataIC50:  15nMAssay Description:Inhibition of mouse JAK1Checked by AuthorMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK1(Mus musculus)
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM26198(4-tert-butyl-15-fluoro-3,5,10-triazatetracyclo[11....)
Affinity DataIC50:  15nMAssay Description:Inhibition of murine Jak 1 protein kinaseMore data for this Ligand-Target Pair