Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
maximum 50k data
Found
1
Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase JAK1' and Ligand = 'BDBM475702'
Target
Tyrosine-protein kinase JAK1
(Homo sapiens (Human))
Leo Pharma
US Patent
Ligand
BDBM475702
(8a-ethyl-7- (7H- pyrrolo[2,3- d]pyrimidin-4- yl)- ...)
Copy SMILES
Affinity Data
EC50: 16nM
Assay Description:
Inhibition of phosphorylation of a synthetic peptide was measured in an HTRF-based assay using the TK substrate-Biotin from the Cisbio HTRFKinEASE TK...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI