Found 2 Enz. Inhib. hit(s) with Target = 'Tyrosyl-DNA phosphodiesterase 1' and Ligand = 'BDBM50232843'
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch Of The Russian Academy Of Sciences
Curated by ChEMBL
Siberian Branch Of The Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured at 1 min interval by fluorimet...More data for this Ligand-Target Pair
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch Of The Russian Academy Of Sciences
Curated by ChEMBL
Siberian Branch Of The Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) assessed as reduction in BHQ1 excision from 3'-end of [32P]-labeled oligonucleotide substrate after 2...More data for this Ligand-Target Pair