Compile Data Set for Download or QSAR
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Found 4 of ic50 for monomerid = 10018
TargetAromatase(Homo sapiens (Human))
University Of Bath

LigandPNGBDBM10018((4-{[(4-cyanophenyl)(4H-1,2,4-triazol-4-yl)amino]m...)
Affinity DataIC50:  12nMpH: 7.5 T: 2°CAssay Description:The extent of in vitro inhibition of aromatase activities was assessed using intact monolayers of JEG-3 cells. Aromatase activity was measured using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Bath

LigandPNGBDBM10018((4-{[(4-cyanophenyl)(4H-1,2,4-triazol-4-yl)amino]m...)
Affinity DataIC50:  12nMpH: 7.5 T: 2°CAssay Description:The extent of in vitro inhibition of aromatase activities was assessed using intact monolayers of JEG-3 cells. Aromatase activity was measured using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Bath

LigandPNGBDBM10018((4-{[(4-cyanophenyl)(4H-1,2,4-triazol-4-yl)amino]m...)
Affinity DataIC50:  40nMAssay Description:The extent of in vitro inhibition of sulfatase activities was assessed using intact monolayers of JEG-3 cells. Sulfatase activity was measured using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Bath

LigandPNGBDBM10018((4-{[(4-cyanophenyl)(4H-1,2,4-triazol-4-yl)amino]m...)
Affinity DataIC50:  40nMpH: 7.5 T: 2°CAssay Description:The extent of in vitro inhibition of sulfatase activities was assessed using intact monolayers of JEG-3 cells. Sulfatase activity was measured using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed