Compile Data Set for Download or QSAR
maximum 50k data
Found 22 of ic50 for monomerid = 119703
TargetHistone deacetylase 6(Homo sapiens (Human))
Universidad Del PaíS Vasco

US Patent
LigandPNGBDBM119703(US8685992, 27)
Affinity DataIC50:  1.60nMT: 2°CAssay Description:The reactions were carried out in a 96-well microplate for fluorometry in a 50 μl reaction volume. After the deacetylation reaction, Fluor-de-Ly...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 6(Homo sapiens (Human))
Universidad Del PaíS Vasco

US Patent
LigandPNGBDBM119703(US8685992, 27)
Affinity DataIC50:  2nMAssay Description:Inhibition of N-terminal GST-tagged full length human HDAC6 expressed in baculovirus expression system in Sf9 cells using AMC-labeled RHKKAc as subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM119703(US8685992, 27)
Affinity DataIC50:  70nMAssay Description:Inhibition of C-terminal GST-tagged full length human HDAC1 expressed in baculovirus expression system in Sf9 cells using AMC-labeled RHKKAc as subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM119703(US8685992, 27)
Affinity DataIC50:  71nMT: 2°CAssay Description:The reactions were carried out in a 96-well microplate for fluorometry in a 50 μl reaction volume. After the deacetylation reaction, Fluor-de-Ly...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 3(Homo sapiens (Human))
Universidad Del PaíS Vasco

US Patent
LigandPNGBDBM119703(US8685992, 27)
Affinity DataIC50:  75nMT: 2°CAssay Description:The reactions were carried out in a 96-well microplate for fluorometry in a 50 μl reaction volume. After the deacetylation reaction, Fluor-de-Ly...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 3(Homo sapiens (Human))
Universidad Del PaíS Vasco

US Patent
LigandPNGBDBM119703(US8685992, 27)
Affinity DataIC50:  80nMAssay Description:Inhibition of C-terminal His-tagged full length human HDAC3 expressed in baculovirus expression system using AMC-labeled RHKKAc as substrate after 2 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Universidad Del PaíS Vasco

US Patent
LigandPNGBDBM119703(US8685992, 27)
Affinity DataIC50:  148nMT: 2°CAssay Description:The reactions were carried out in a 96-well microplate for fluorometry in a 50 μl reaction volume. After the deacetylation reaction, Fluor-de-Ly...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 8(Homo sapiens (Human))
Universidad Del PaíS Vasco

US Patent
LigandPNGBDBM119703(US8685992, 27)
Affinity DataIC50:  150nMAssay Description:Inhibition of full length human HDAC8 expressed in an E. coli expression system using AMC-labeled RHKAcKAc as substrate after 2 hrs by fluorescence a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universidad Del PaíS Vasco

US Patent
LigandPNGBDBM119703(US8685992, 27)
Affinity DataIC50:  157nMT: 2°CAssay Description:The reactions were carried out in a 96-well microplate for fluorometry in a 50 μl reaction volume. After the deacetylation reaction, Fluor-de-Ly...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 2(Homo sapiens (Human))
Universidad Del PaíS Vasco

US Patent
LigandPNGBDBM119703(US8685992, 27)
Affinity DataIC50:  160nMAssay Description:Inhibition of C-terminal His-tagged full length human HDAC2 expressed in baculovirus expression system in Sf9 cells using AMC-labeled RHKKAc as subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 9(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM119703(US8685992, 27)
Affinity DataIC50:  160nMAssay Description:Inhibition of C-terminal His-tagged human HDAC9 (604 to 1066 residues) expressed in baculovirus expression system after 2 hrs by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 9(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM119703(US8685992, 27)
Affinity DataIC50:  163nMT: 2°CAssay Description:The reactions were carried out in a 96-well microplate for fluorometry in a 50 μl reaction volume. After the deacetylation reaction, Fluor-de-Ly...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 5(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM119703(US8685992, 27)
Affinity DataIC50:  220nMAssay Description:Inhibition of N-terminal GST-tagged full length human HDAC5 expressed in baculovirus expression system in Sf9 cells using AMC-labeled RHKKAc as subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM119703(US8685992, 27)
Affinity DataIC50:  222nMT: 2°CAssay Description:The reactions were carried out in a 96-well microplate for fluorometry in a 50 μl reaction volume. After the deacetylation reaction, Fluor-de-Ly...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 7(Homo sapiens (Human))
Universidad Del PaíS Vasco

US Patent
LigandPNGBDBM119703(US8685992, 27)
Affinity DataIC50:  290nMT: 2°CAssay Description:The reactions were carried out in a 96-well microplate for fluorometry in a 50 μl reaction volume. After the deacetylation reaction, Fluor-de-Ly...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 7(Homo sapiens (Human))
Universidad Del PaíS Vasco

US Patent
LigandPNGBDBM119703(US8685992, 27)
Affinity DataIC50:  290nMAssay Description:Inhibition of N-terminal GST-tagged human HDAC7 (518 to end residues) expressed in baculovirus expression system using AMC-labeled RHKKAc as substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine deacetylase HDAC10(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM119703(US8685992, 27)
Affinity DataIC50:  290nMAssay Description:Inhibition of N-terminal GST-tagged human HDAC10 (1 to 631 residues) expressed in baculovirus expression system in Sf9 cells RHKAcKAc after 2 hrs by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine deacetylase HDAC10(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM119703(US8685992, 27)
Affinity DataIC50:  294nMT: 2°CAssay Description:The reactions were carried out in a 96-well microplate for fluorometry in a 50 μl reaction volume. After the deacetylation reaction, Fluor-de-Ly...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 11(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM119703(US8685992, 27)
Affinity DataIC50:  340nMAssay Description:Inhibition of N-terminal GST-tagged human HDAC11 expressed in baculovirus expression systemRHKAcKAc after 2 hrs by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 11(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM119703(US8685992, 27)
Affinity DataIC50:  341nMT: 2°CAssay Description:The reactions were carried out in a 96-well microplate for fluorometry in a 50 μl reaction volume. After the deacetylation reaction, Fluor-de-Ly...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 4(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM119703(US8685992, 27)
Affinity DataIC50:  1.08E+3nMAssay Description:Inhibition of N-terminal GST-tagged human HDAC4 (627 to 1085 residues) expressed in baculovirus expression system using AMC-labeled RHKKAc as substra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM119703(US8685992, 27)
Affinity DataIC50:  1.08E+3nMT: 2°CAssay Description:The reactions were carried out in a 96-well microplate for fluorometry in a 50 μl reaction volume. After the deacetylation reaction, Fluor-de-Ly...More data for this Ligand-Target Pair
In DepthDetails US Patent