Compile Data Set for Download or QSAR
maximum 50k data
Found 13 of ec50 for monomerid = 43363
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Pcmd

Curated by PubChem BioAssay
LigandPNGBDBM43363(2,5-bis(chloranyl)-3-piperidin-1-yl-6-(2-piperidin...)
Affinity DataEC50:  2.42E+3nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 7(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM43363(2,5-bis(chloranyl)-3-piperidin-1-yl-6-(2-piperidin...)
Affinity DataEC50:  830nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 19(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM43363(2,5-bis(chloranyl)-3-piperidin-1-yl-6-(2-piperidin...)
Affinity DataEC50:  670nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 16(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM43363(2,5-bis(chloranyl)-3-piperidin-1-yl-6-(2-piperidin...)
Affinity DataEC50:  1.65E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMatrix metalloproteinase-14 [1-36](Homo sapiens (Human))
Sanford-Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM43363(2,5-bis(chloranyl)-3-piperidin-1-yl-6-(2-piperidin...)
Affinity DataEC50:  4.53E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM43363(2,5-bis(chloranyl)-3-piperidin-1-yl-6-(2-piperidin...)
Affinity DataEC50:  1.14E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 19(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM43363(2,5-bis(chloranyl)-3-piperidin-1-yl-6-(2-piperidin...)
Affinity DataEC50:  82nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 4(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM43363(2,5-bis(chloranyl)-3-piperidin-1-yl-6-(2-piperidin...)
Affinity DataEC50:  1.82E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 4(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM43363(2,5-bis(chloranyl)-3-piperidin-1-yl-6-(2-piperidin...)
Affinity DataEC50:  269nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 7(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM43363(2,5-bis(chloranyl)-3-piperidin-1-yl-6-(2-piperidin...)
Affinity DataEC50:  158nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 16(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM43363(2,5-bis(chloranyl)-3-piperidin-1-yl-6-(2-piperidin...)
Affinity DataEC50:  121nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetRegulator of G-protein signaling 8(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM43363(2,5-bis(chloranyl)-3-piperidin-1-yl-6-(2-piperidin...)
Affinity DataEC50:  78nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Pcmd

Curated by PubChem BioAssay
LigandPNGBDBM43363(2,5-bis(chloranyl)-3-piperidin-1-yl-6-(2-piperidin...)
Affinity DataEC50:  2.32E+3nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Brent Stockwell, Columbia University ML...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay