Compile Data Set for Download or QSAR
maximum 50k data
Found 29 of ki for monomerid = 50001450
TargetSubstance-P receptor(Rattus norvegicus (rat))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  0.0420nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  0.0440nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  0.0540nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  0.0590nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtachykinin-1(Homo sapiens (Human))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtachykinin-1(RAT)
National Institutes Of Health

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance P(GUINEA PIG)
National Institutes Of Health

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  0.240nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtachykinin-1(MOUSE)
National Institutes Of Health

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  0.310nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  0.330nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  1.02nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  1.10nMAssay Description:Ability to inhibit the binding of [125I]physalaemin to the SP receptors in rat telencephalon slicesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  1.60nMAssay Description:Compound was evaluated for affinity towards human tachykinin NK-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  2.80nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetEledoisin(Eledone moschata (Musky octopus) (Ozaena moschata))
National Institutes Of Health

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  19nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetATP synthase subunit a(RAT)
National Institutes Of Health

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  21nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetClass E basic helix-loop-helix protein 22(MOUSE)
National Institutes Of Health

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  47nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  51nMAssay Description:Evaluated for the binding affinity against NK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  102nMAssay Description:The compound was tested for competition binding with [3H]NKA against the CHO cells from cloned human Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP synthase subunit a(RAT)
National Institutes Of Health

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  106nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtachykinin-1(RAT)
National Institutes Of Health

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  112nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtachykinin-1(MOUSE)
National Institutes Of Health

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  125nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  129nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-K receptor(GUINEA PIG)
National Institutes Of Health

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  200nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  1.29E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProthrombin(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1/A2a/A2b/A3(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi: >3.00E+4nMAssay Description:Ability to inhibit the binding of [3H]N6-phenylisopropyl adenosine to adenosine receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed