Affinity DataEC50: 7.80nMAssay Description:Agonist activity at recombinant human MOR expressed in CHO cell membranes after 60 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Binding affinity to rat brain opioid receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 250nMAssay Description:Binding affinity to opiate receptor in rat brain homogenatesMore data for this Ligand-Target Pair