Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataIC50: 2.90nMAssay Description:Binding affinity towards 5-HT2C receptor from rat using [3H]-mesulergine as radioligandMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
University Of GöTeborg
Curated by ChEMBL
University Of GöTeborg
Curated by ChEMBL
Affinity DataIC50: 2.90nMAssay Description:Inhibition of [3H]-mesulergine binding to 5-hydroxytryptamine 2C receptor in rat brain membranesMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibitory binding of [3H]-pirenzepine to human Muscarinic acetylcholine receptor M1 in membranes from CHO-K1 cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of binding of 1.0 nM [3H]-pirenzepine to cloned human Muscarinic acetylcholine receptor M1 expressed in membranes from CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Binding affinity towards D1 CNS receptor of rat corpus striatum using [3H]-SCH-23,390 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibitory binding of [3H]-SCH-23,390 to Dopamine receptor D1 in membranes from rat corpus striatumMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of [3H]-ketanserin binding to 5-hydroxytryptamine 2A receptor from rat brainMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor from rat frontal cortex using [3H]-ketanserin as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Binding affinity towards Dopamine receptor D2 of rat corpus striatum using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibitory binding of [3H]-spiperone to Dopamine receptor D2 in membranes from rat corpus striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Tested in vitro for its ability to displace 3[H] clozapine from Muscarinic acetylcholine receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Binding affinity towards human Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:Binding affinity was determined against Muscarinic acetylcholine receptor using [3H]QNB as radioligand in rat brain.More data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:Binding activity against muscarinic receptor in rat brain using [3H]QNB as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Binding activity against dopamine D1 receptor in rat brain, using [3H]-SCH-23,390 as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Binding affinity against Dopamine receptor D1 using [3H]-SCN 23390 in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Binding affinity towards human D4.2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Binding affinity towards human Dopamine receptor D3More data for this Ligand-Target Pair
Affinity DataIC50: 218nMAssay Description:Binding activity against Dopamine receptor D2 in rat brain, using [3H]-Spiperone as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 218nMAssay Description:Binding affinity for Dopamine receptor D2 using [3H]-spiperone in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 758nMAssay Description:Displacement of 3[H]spiroperidol from Dopamine receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 758nMAssay Description:Relative affinity for dopamine receptor by displacement of [3H]spiroperidol (2.2 nM) from (in vitro) dopamine binding sites in rat caudate nucleiMore data for this Ligand-Target Pair