TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania
Curated by PDSP Ki Database
University Of Pennsylvania
Curated by PDSP Ki Database
Affinity DataKi: 1.10nMAssay Description:Displacement of radiolabeled DPDPE-Cl from delta opioid receptor in Hartley guinea pig brainMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(MOUSE)
Memorial Sloan-Kettering Cancer Center
Curated by PDSP Ki Database
Memorial Sloan-Kettering Cancer Center
Curated by PDSP Ki Database
TargetMu-type opioid receptor(MOUSE)
Memorial Sloan-Kettering Cancer Center
Curated by PDSP Ki Database
Memorial Sloan-Kettering Cancer Center
Curated by PDSP Ki Database
Affinity DataKi: 2nMAssay Description:Displacement of [3H]diprenorphine from human cloned delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:Displacement of radiolabeled DAMGO from mu opioid receptor in Hartley guinea pig brainMore data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Inhibition of [3H]-DTLET binding torat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania
Curated by PDSP Ki Database
University Of Pennsylvania
Curated by PDSP Ki Database
Affinity DataKi: 19nMAssay Description:Displacement of [3H]diprenorphine from human cloned mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Compound was evaluated for binding affinity towards mu-specific opiate receptor from combinatorial peptoid libraryMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Inhibition of [3H]-DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
TargetOprd1b protein(Danio rerio)
Instituto De Qu£Mica Avanzada De Catalu£A (Iqac-Csic)
Curated by ChEMBL
Instituto De Qu£Mica Avanzada De Catalu£A (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 45nMAssay Description:Displacement of [3H]DPN from zebrafish delta 1b opioid receptor expressed in HEK293 cell membranes after 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 277nMAssay Description:Displacement of radiolabeled NalBzOH from kappa3 opioid receptor in Hartley guinea pig brainMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Danio rerio)
Instituto De Qu£Mica Avanzada De Catalu£A (Iqac-Csic)
Curated by ChEMBL
Instituto De Qu£Mica Avanzada De Catalu£A (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 684nMAssay Description:Displacement of [3H]DPN from zebrafish mu opioid receptor expressed in HEK293 cell membranes after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania
Curated by PDSP Ki Database
University Of Pennsylvania
Curated by PDSP Ki Database
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Kentucky
Curated by ChEMBL
University Of Kentucky
Curated by ChEMBL
Affinity DataKi: 4.47E+3nMAssay Description:Displacement of radiolabeled U69593 from kappa1 opioid receptor in Hartley guinea pig brainMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania
Curated by PDSP Ki Database
University Of Pennsylvania
Curated by PDSP Ki Database
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]diprenorphine from human cloned kappa opioid receptorMore data for this Ligand-Target Pair