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Found 8 of ki for monomerid = 50021959
TargetBeta-lactamase TEM(Escherichia coli)
Cnrs-Cercoa

Curated by ChEMBL
LigandPNGBDBM50021959(CHEMBL777 | MM 14151 | US9120808, Clavulanic acid ...)
Affinity DataKi:  800nMAssay Description:Inhibition constant (Ki) for TEM-1 beta-lactamaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase SHV-1(Klebsiella pneumoniae (Enterobacteria))
Case Western Reserve University

LigandPNGBDBM50021959(CHEMBL777 | MM 14151 | US9120808, Clavulanic acid ...)
Affinity DataKi:  2.00E+3nM IC50:  100nMpH: 7.4Assay Description:Steady state kinetics were performed on an Agilent 8453 diode array spectrophotometer in 10 mM phosphate-buffered saline (pH 7.4). IC50, defined as t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Mycobacterium tuberculosis H37Rv)
Indian Institute Of Technology

LigandPNGBDBM50021959(CHEMBL777 | MM 14151 | US9120808, Clavulanic acid ...)
Affinity DataKi:  6.30E+3nMpH: 7.2Assay Description:Steady state kinetics were performed on an Agilent 8453 diode array spectrophotometer in sodium phosphate buffer (50 mM, pH 7.2) and a 1 cm pathlengt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Escherichia coli)
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM50021959(CHEMBL777 | MM 14151 | US9120808, Clavulanic acid ...)
Affinity DataKi:  1.10E+4nMAssay Description:Inhibition of Klebsiella pneumoniae 1534 beta-lactamase KPC-2 by competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase SHV-5(Klebsiella pneumoniae)TBA
LigandPNGBDBM50021959(CHEMBL777 | MM 14151 | US9120808, Clavulanic acid ...)
Affinity DataKi:  2.54E+4nMAssay Description:Inhibition of Klebsiella pneumoniae beta-lactamase SHV-105More data for this Ligand-Target Pair
In DepthDetails Article
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50021959(CHEMBL777 | MM 14151 | US9120808, Clavulanic acid ...)
Affinity DataKi:  1.08E+5nMAssay Description:Inhibition of Citrobacter freundii beta-lactamase SHV-95More data for this Ligand-Target Pair
In DepthDetails Article
TargetBeta-lactamase(Acinetobacter baumannii)TBA
LigandPNGBDBM50021959(CHEMBL777 | MM 14151 | US9120808, Clavulanic acid ...)
Affinity DataKi:  2.27E+5nMAssay Description:Inhibition of Acinetobacter baumannii beta-lactamase SHV-48More data for this Ligand-Target Pair
In DepthDetails Article
TargetBeta-lactamase SHV-1(Klebsiella pneumoniae (Enterobacteria))
Case Western Reserve University

LigandPNGBDBM50021959(CHEMBL777 | MM 14151 | US9120808, Clavulanic acid ...)
Affinity DataKi:  2.29E+5nMAssay Description:Inhibition of Klebsiella pneumoniae beta-lactamase SHV-89More data for this Ligand-Target Pair
In DepthDetails Article