Affinity DataKi: 800nMAssay Description:Inhibition constant (Ki) for TEM-1 beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nM IC50: 100nMpH: 7.4Assay Description:Steady state kinetics were performed on an Agilent 8453 diode array spectrophotometer in 10 mM phosphate-buffered saline (pH 7.4). IC50, defined as t...More data for this Ligand-Target Pair
Affinity DataKi: 6.30E+3nMpH: 7.2Assay Description:Steady state kinetics were performed on an Agilent 8453 diode array spectrophotometer in sodium phosphate buffer (50 mM, pH 7.2) and a 1 cm pathlengt...More data for this Ligand-Target Pair
Affinity DataKi: 1.10E+4nMAssay Description:Inhibition of Klebsiella pneumoniae 1534 beta-lactamase KPC-2 by competitive assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.54E+4nMAssay Description:Inhibition of Klebsiella pneumoniae beta-lactamase SHV-105More data for this Ligand-Target Pair
Affinity DataKi: 1.08E+5nMAssay Description:Inhibition of Citrobacter freundii beta-lactamase SHV-95More data for this Ligand-Target Pair
Affinity DataKi: 2.27E+5nMAssay Description:Inhibition of Acinetobacter baumannii beta-lactamase SHV-48More data for this Ligand-Target Pair
Affinity DataKi: 2.29E+5nMAssay Description:Inhibition of Klebsiella pneumoniae beta-lactamase SHV-89More data for this Ligand-Target Pair