TargetDelta-type opioid receptor(MOUSE)
C.N.R. Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
C.N.R. Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
Affinity DataKi: 0.710nMAssay Description:Displacement of [3H]DPDPE from mouse brain delta opioid receptor by scintillation counting analysisMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
C.N.R. Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
C.N.R. Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]diprenorphine from human delta opioid receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]DPDPE from DOR in Sprague-Dawley rat brain membranes after 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]-deltorphine from human delta opioid receptor expressed in CHO-K1 cells by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]-DPDPE from DOR in rat brain membranes measured by competitive radioligand receptor binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Inhibitory activity against Opioid receptor delta 1 in rat brain membranes using [3H]-DADLE as a radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 1.57nMAssay Description:Affinity of [H]DADLE to the delta opioid receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Compound was evaluated for binding affinity towards Opioid receptor delta 1 by displacement of [3H]-DADLE radioligandMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
C.N.R. Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
C.N.R. Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Binding affinity towards opioid Delta receptor using [3H]DADLE as radioligandMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
C.N.R. Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
C.N.R. Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Binding affinity towards opioid Delta receptor using [3H]DADLE as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]deltorphine 2 from human delta opioid receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Inhibition of [3H]-DPDPE radioligand binding to rat opioid receptor delta 1 site from rat brain membranesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
C.N.R. Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
C.N.R. Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Binding affinity against Opioid receptor delta 1 using [3H][D-Ala2, D-Leu5]-enkephalin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Binding affinity for delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Inhibition of binding of [3H]-DPDPE to opioid receptor delta 1 from rat brain membrane.More data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]DADLE from delta opioid receptor in rat brain after 60 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:In vitro binding affinity to Opioid receptor delta 1 in rat brain membranes by [3H]DADLE (Tyr-D-Ala-Gly-Phe-D-Leu) displacement.More data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:Binding affinity at opioid receptor delta 1 by displacement of [3H]DADLE in rat brain membraneMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
C.N.R. Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
C.N.R. Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
Affinity DataKi: 16.6nMAssay Description:Displacement of [3H]-DPDPE from mouse DOR expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 352nMAssay Description:Displacement of [125I]FK33824 from human cloned mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 695nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University
Curated by ChEMBL
Kitasato University
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum membraneMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 1.30E+3nMAssay Description:Inhibition of binding of [3H]DAMGO to opioid receptor mu 1 from rat brain membrane.More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 1.30E+3nMAssay Description:Binding affinity of the compound was determined by inhibition of [3H]-DAMGO binding to Opioid receptor mu 1 from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Binding affinity against Opioid receptor mu 1 using [3H][D-Ala2, MePhe4, Gly-ol5]-enkephalin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Binding affinity for mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.35E+3nMAssay Description:Binding affinity against Opioid receptor kappa 1 using [3H]-U-69,593 as radioligandMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 1.61E+3nMAssay Description:Binding affinity towards opioid Mu receptor using [3H]DAMGO as radioligandMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 1.61E+3nMAssay Description:Compound was evaluated for binding affinity towards Opioid receptor mu 1 by displacement of [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 1.61E+3nMAssay Description:Affinity of [3H]DAMGO to the mu opioid receptor from rat brainMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 1.61E+3nMAssay Description:Binding affinity towards opioid Mu receptor using [3H]DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.38E+3nMAssay Description:Displacement of [3H]DAMGO from mouse brain mu opioid receptor by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.75E+3nMAssay Description:Displacement of [3H]U-69,593 from mouse brain kappa opioid receptor by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.54E+3nMAssay Description:Binding affinity towards opioid kappa receptor using [3H]U-69593 as radioligandMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University
Curated by ChEMBL
Kitasato University
Curated by ChEMBL
Affinity DataKi: 3.54E+3nMAssay Description:Compound was evaluated for binding affinity towards Opioid receptor kappa 1 by displacement of [3H]-U-69,593 radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.54E+3nMAssay Description:Binding affinity towards opioid kappa receptor using [3H]U-69593 as radioligandMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 3.54E+3nMAssay Description:Affinity of [3H]U-69593 to opioid receptor kappa 1 from rat brainMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 3.97E+3nMAssay Description:In vitro radioligand binding assay, for inhibition of [3H]DAMGO (Tyr-D-Ala-Gly-(Me)-Phe-Gly-ol) binding to Opioid receptor mu 1 in rat brain membrane...More data for this Ligand-Target Pair
Affinity DataKi: 4.17E+3nMAssay Description:Displacement of [125I]D-pro10-dynorphin from human cloned kappa opioid receptorMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 8.07E+3nMAssay Description:Binding affinity at Opioid receptor mu 1 by displacement of [3H]DAMGO in rat brain membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University
Curated by ChEMBL
Kitasato University
Curated by ChEMBL
Affinity DataKi: 8.76E+3nMAssay Description:Binding affinity at Opioid receptor kappa 1 by displacement of [3H]U-69593 in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University
Curated by ChEMBL
Kitasato University
Curated by ChEMBL
Affinity DataKi: 1.17E+4nMAssay Description:In vitro radioligand binding assay, for inhibition of [3H]U-69593 binding to Opioid receptor kappa 1, in guinea pig brain membranes.More data for this Ligand-Target Pair