Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ic50 for monomerid = 50053929
TargetAdenosine receptor A3(Homo sapiens (Human))
National And Kapodistrian University Of Athens

Curated by ChEMBL
LigandPNGBDBM50053929(CHEMBL88147 | N-(9-Chloro-2-furan-2-yl-[1,2,4]tria...)
Affinity DataIC50:  0.0977nMAssay Description:Antagonist activity at wild type A3R (unknown origin) expressed in Flp-In-CHO cells assessed as inhibition of NECA reduced forskolin stimulated cAMP ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
National And Kapodistrian University Of Athens

Curated by ChEMBL
LigandPNGBDBM50053929(CHEMBL88147 | N-(9-Chloro-2-furan-2-yl-[1,2,4]tria...)
Affinity DataIC50:  7.20nMAssay Description:Antagonist activity at human adenosine A3 receptor expressed in CHO cells by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
National And Kapodistrian University Of Athens

Curated by ChEMBL
LigandPNGBDBM50053929(CHEMBL88147 | N-(9-Chloro-2-furan-2-yl-[1,2,4]tria...)
Affinity DataIC50:  48nMAssay Description:Antagonist activity at wild type A1R (unknown origin) expressed in CHO-K1 cells assessed as inhibition of NECA reduced forskolin stimulated cAMP accu...More data for this Ligand-Target Pair
In DepthDetails PubMed