Compile Data Set for Download or QSAR
maximum 50k data
Found 40 of ki for monomerid = 50158610
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi:  0.270nMAssay Description:In vitro binding affinity was determined as displacement of [3H]N-R-methylhistamine from C6 cell membranes expressing human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi:  1nMAssay Description:In vitro binding affinity was determined as displacement of [3H]N-R-methylhistamine from C6 cell membranes expressing rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity to human H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi:  204nMAssay Description:Binding affinity to human recombinant M3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi:  351nMAssay Description:Binding affinity to human recombinant M4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi:  432nMAssay Description:Binding affinity to human recombinant 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi:  437nMAssay Description:Binding affinity to human recombinant M5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi:  462nMAssay Description:Binding affinity to human recombinant M2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi:  1.71E+3nMAssay Description:Binding affinity to human recombinant H2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi:  2.72E+3nMAssay Description:Binding affinity to human recombinant 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi:  3.15E+3nMAssay Description:Binding affinity to human recombinant 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi:  3.27E+3nMAssay Description:Binding affinity to human recombinant M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi:  5.44E+3nMAssay Description:Binding affinity to human recombinant H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi:  6.38E+3nMAssay Description:Binding affinity to human recombinant 5HT1D receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant alpha1A adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant alpha1B adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant alpha1D adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant alpha2A adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant alpha2C adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant beta3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant Dopamine D1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant Dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant Dopamine D3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant Dopamine D5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant beta1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant 5HT7 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant 5HT6 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant 5HT5A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant 5HT3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant 5HT1E receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant DATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant 5HT1B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant H4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant Dopamine D4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant SERTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant sigma1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant alpha2B adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50158610((4-Fluoro-phenyl)-{2-[2-((R)-2-methyl-pyrrolidin-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant beta2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed