TargetSerine/threonine-protein kinase SIK3 [59-1321](Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 120nMAssay Description:Binding affinity to QSKMore data for this Ligand-Target Pair
Affinity DataKd: 200nMAssay Description:Binding affinity to PIM1More data for this Ligand-Target Pair
Affinity DataKd: 80nMAssay Description:Binding affinity to DAPK1More data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 47nMAssay Description:Binding affinity to CAMK1DMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 350nMAssay Description:Binding affinity to PIK3CGMore data for this Ligand-Target Pair
Affinity DataKd: 1.30E+3nMAssay Description:Binding affinity to PFTAIRE2More data for this Ligand-Target Pair
Affinity DataKd: 4.00E+3nMAssay Description:Binding affinity to NEK7More data for this Ligand-Target Pair
Affinity DataKd: 62nMAssay Description:Binding affinity to RPS6KA4(Kin.Dom.1-N-terminal)More data for this Ligand-Target Pair
TargetSTE20-like serine/threonine-protein kinase(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 8.5nMAssay Description:Binding affinity to FLT3More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to EPHB4More data for this Ligand-Target Pair
Affinity DataKd: 98nMAssay Description:Binding affinity to EPHB6More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 6.10nMAssay Description:Binding affinity to IRAK1More data for this Ligand-Target Pair
Affinity DataKd: 1.80nMAssay Description:Binding affinity to PKN2More data for this Ligand-Target Pair
Affinity DataKd: 3.40nMAssay Description:Binding affinity to DRAK1More data for this Ligand-Target Pair
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 110nMAssay Description:Binding affinity to CSF1RMore data for this Ligand-Target Pair
Affinity DataKd: 160nMAssay Description:Binding affinity to PRKCEMore data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to RIPK1More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 15(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 3.40nMAssay Description:Binding affinity to MAP3K15More data for this Ligand-Target Pair
Affinity DataKd: 490nMAssay Description:Binding affinity to LTKMore data for this Ligand-Target Pair
Affinity DataKd: 210nMAssay Description:Binding affinity to CHEK2More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor Tie-1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 680nMAssay Description:Binding affinity to TIE1More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 4.40E+3nMAssay Description:Binding affinity to AKT1More data for this Ligand-Target Pair
Affinity DataKd: 43nMAssay Description:Binding affinity to PAK2More data for this Ligand-Target Pair
Affinity DataKd: 5.90E+3nMAssay Description:Binding affinity to YANK2More data for this Ligand-Target Pair
Affinity DataKd: 380nMAssay Description:Binding affinity to EPHA1More data for this Ligand-Target Pair
TargetMuscle, skeletal receptor tyrosine-protein kinase(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to MUSKMore data for this Ligand-Target Pair
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 1.10E+3nMAssay Description:Binding affinity to STK39More data for this Ligand-Target Pair
TargetMyosin light chain kinase, smooth muscle(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 12nMAssay Description:Binding affinity to MLCKMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 4(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 23nMAssay Description:Binding affinity to MAP4K4More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CSNK1G1More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CDK8More data for this Ligand-Target Pair
Affinity DataKd: 1nMAssay Description:Binding affinity to LATS2More data for this Ligand-Target Pair
Affinity DataKd: 1.10E+3nMAssay Description:Binding affinity to EGFRMore data for this Ligand-Target Pair
Affinity DataKd: 28nMAssay Description:Binding affinity to RPS6KA1(Kin.Dom.1-N-terminal)More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CDK11More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 9nMAssay Description:Binding affinity to IKK-alphaMore data for this Ligand-Target Pair
Affinity DataKd: 1.70E+3nMAssay Description:Binding affinity to BRKMore data for this Ligand-Target Pair
TargetBone morphogenetic protein receptor type-1B(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 57nMAssay Description:Binding affinity to BMPR1BMore data for this Ligand-Target Pair
Affinity DataKd: 1.00E+3nMAssay Description:Binding affinity to ULK1More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 6.60nMAssay Description:Binding affinity to TNK2More data for this Ligand-Target Pair
TargetAnkyrin repeat and protein kinase domain-containing protein 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 32nMAssay Description:Binding affinity to ANKK1More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 20(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to ZAKMore data for this Ligand-Target Pair
Affinity DataKd: 2.50E+3nMAssay Description:Binding affinity to ACVR2AMore data for this Ligand-Target Pair
Affinity DataKd: 230nMAssay Description:Binding affinity to METMore data for this Ligand-Target Pair
Affinity DataKd: 13nMAssay Description:Binding affinity to SRPK3More data for this Ligand-Target Pair
Affinity DataKd: 200nMAssay Description:Binding affinity to SBK1More data for this Ligand-Target Pair
Affinity DataKd: 14nMAssay Description:Binding affinity to MARK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MRCK beta(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 1.00E+3nMAssay Description:Binding affinity to MRCKBMore data for this Ligand-Target Pair