TargetDual specificity protein phosphatase 5 [180-384](Homo sapiens (Human))
Texas Wesleyan University
Texas Wesleyan University
Affinity DataKi: 25nM ΔG°: -10.4kcal/mole IC50: 4.40E+4nMT: 2°CAssay Description:For the 96-well plate validation assay, sodium orthovanadate (Sigma Aldrich) was utilized as a positive control for inhibition [Swarup et al., Bioche...More data for this Ligand-Target Pair
TargetNucleoside triphosphate diphosphohydrolase 3(Rattus norvegicus)
University Of Bonn
Curated by ChEMBL
University Of Bonn
Curated by ChEMBL
Affinity DataKi: 1.27E+4nMAssay Description:Inhibition of rat recombinant NTPDase3 expressed in CHO cellsMore data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 2(Rattus norvegicus)
University Of Bonn
Curated by ChEMBL
University Of Bonn
Curated by ChEMBL
Affinity DataKi: 6.54E+4nMAssay Description:Inhibition of rat NTPDase 2More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 2(Rattus norvegicus)
University Of Bonn
Curated by ChEMBL
University Of Bonn
Curated by ChEMBL
Affinity DataKi: 6.54E+4nMAssay Description:Inhibition of rat recombinant NTPDase2 expressed in CHO cellsMore data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 8(Homo sapiens (Human))
University Of Bonn
Curated by ChEMBL
University Of Bonn
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human NTPDase 8 expressed in COS7 cellsMore data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rattus norvegicus)
University Of Bonn
Curated by ChEMBL
University Of Bonn
Curated by ChEMBL
Affinity DataKi: 3.00E+5nMAssay Description:Inhibition of rat NTPDase 1More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rattus norvegicus)
University Of Bonn
Curated by ChEMBL
University Of Bonn
Curated by ChEMBL
Affinity DataKi: 3.00E+5nMAssay Description:Inhibition of rat recombinant NTPDase1 expressed in CHO cellsMore data for this Ligand-Target Pair