TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
George Washington University Medical Center
Curated by ChEMBL
George Washington University Medical Center
Curated by ChEMBL
Affinity DataKd: 38.2nMAssay Description:Binding affinity against MCF cells in the membrane preparation using radioligand binding assay.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
George Washington University Medical Center
Curated by ChEMBL
George Washington University Medical Center
Curated by ChEMBL
Affinity DataKd: 11.6nMAssay Description:Binding constant (Kd) for [3H]DTG binding to Sigma opioid receptor type 1 of guinea pig brain membranes at 5 uM BNITMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
George Washington University Medical Center
Curated by ChEMBL
George Washington University Medical Center
Curated by ChEMBL
Affinity DataKd: 13.6nMAssay Description:Binding constant (Kd) for [3H]DTG binding to Sigma opioid receptor type 1 of guinea pig brain membranes at 1 uM BNITMore data for this Ligand-Target Pair