Affinity DataIC50: 0.260nMAssay Description:Inhibition of [3H]-mepyramine binding to the histamine receptor in guinea pig cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inhibition of guinea pig histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.58nMAssay Description:Potency against histamine H1 receptor on guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Inhibition of [3H]-mepyramine binding to the histamine receptor in guinea pig cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 6.10nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 6.90nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 7.40nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibitory activity of the compound against Tritiated [3H]- mepyramine binding to histamine H1 receptor in guinea pig cerebral cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 8.40nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 8.40nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 8.60nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 8.80nMAssay Description:Inhibition of [3H]-mepyramine binding to the Histamine H1 receptor in guinea pig cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibitory activity of the compound against Tritiated [3H]- mepyramine binding to Histamine H1 receptor in guinea pig cerebral cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 9.10nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 9.90nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:In vitro antagonistic activity at the Histamine H1 receptor in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:In vitro antagonistic activity at the Histamine H1 receptor in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:In vitro antagonistic activity at the Histamine H1 receptor in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Inhibition of [3H]-mepyramine binding to the Histamine H1 receptor in guinea pig cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:In vitro antagonistic activity at the Histamine H1 receptor in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:In vitro antagonistic activity at the Histamine H1 receptor in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Displacement of [3H]mepyramine from histamine H1 receptor in guinea pig cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of [3H]-mepyramine binding to the histamine receptor in guinea pig cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Displacement of [3H]mepyramine from histamine H1 receptor in guinea pig cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:In vitro antagonistic activity at the Histamine H1 receptor in guinea pig ileumMore data for this Ligand-Target Pair