BindingDB PrimarySearch

Found 68 of kd for UniProtKB: P31389

Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM22567(3H]pyrilamine | CHEMBL511 | Dorantamin | Mepyramin...)

Kd: 0.851nMAssay Description:Antagonist activity at H1R in guinea pig ileum assessed as inhibition of histamine-induced muscle contraction after 15 minsMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM24226(1-[(4-fluorophenyl)methyl]-N-{1-[2-(4-methoxypheny...)

Kd: 3.80nMAssay Description:Antagonist activity at H1R in guinea pig ileum assessed as inhibition of histamine-induced muscle contraction after 15 minsMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50419322(CHEMBL1910386)

Kd: 3.80nMAssay Description:Antagonist activity at H1R in guinea pig ileum assessed as inhibition of histamine-induced muscle contraction after 15 minsMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50419326(CHEMBL1910381)

Kd: 4.90nMAssay Description:Antagonist activity at H1R in guinea pig ileum assessed as inhibition of histamine-induced muscle contraction after 15 minsMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50031679(7-[3-(4-Benzhydrylidene-piperidin-1-yl)-propoxy]-2...)

Kd: 5.90nMAssay Description:dissociation constant was determined against H1 receptor of guinea pig lung membranes using radioligand binding assays.More data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50031686(6-[3-(4-Benzhydrylidene-piperidin-1-yl)-propoxy]-4...)

Kd: 6nMAssay Description:Dissociation constant was determined against H1 receptor of guinea pig lung membranes using radioligand binding assays.More data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50419327(CHEMBL1910380)

Kd: 7.24nMAssay Description:Antagonist activity at H1R in guinea pig ileum assessed as inhibition of histamine-induced muscle contraction after 15 minsMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50419325(CHEMBL1910382)

Kd: 7.59nMAssay Description:Antagonist activity at H1R in guinea pig ileum assessed as inhibition of histamine-induced muscle contraction after 15 minsMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50419324(CHEMBL1910384)

Kd: 8.51nMAssay Description:Antagonist activity at H1R in guinea pig ileum assessed as inhibition of histamine-induced muscle contraction after 15 minsMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50419329(CHEMBL1910378)

Kd: 10.7nMAssay Description:Antagonist activity at H1R in guinea pig ileum assessed as inhibition of histamine-induced muscle contraction after 15 minsMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50017674((2-Benzhydryloxy-ethyl)-dimethyl-amine | 2-(benzhy...)

Kd: 11.8nMAssay Description:Antagonist activity at H1R in guinea pig ileum assessed as inhibition of histamine-induced muscle contraction after 15 minsMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50419323(CHEMBL1910385)

Kd: 12.6nMAssay Description:Antagonist activity at H1R in guinea pig ileum assessed as inhibition of histamine-induced muscle contraction after 15 minsMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50419328(CHEMBL1910379)

Kd: 20.4nMAssay Description:Antagonist activity at H1R in guinea pig ileum assessed as inhibition of histamine-induced muscle contraction after 15 minsMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM86171(Arpromidine | CAS_65895 | NSC_65895)

Kd: 22.4nMAssay Description:Antagonist activity at histamine H1 receptor in guinea pig ileum assessed as inhibition of histamine-induced positive chronotropic activityMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50017376((+/-)1-(4-tert-butylphenyl)-4-(4-(hydroxydiphenylm...)

Kd: 35nMAssay Description:Dissociation constant was determined against H1 receptor of guinea pig lung membranes using radioligand binding assays.More data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50421337(CHEMBL432527)

Kd: 214nMAssay Description:Inhibition of specific binding of [3H]mepyramine to Histamine 1 receptors in guinea-pigMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50411492(CHEMBL394144)

Kd: >251nMAssay Description:Antagonist activity at histamine H1 receptor in guinea pig ileum assessed as inhibition of histamine-induced longitudinal smooth muscle contractionMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50017376((+/-)1-(4-tert-butylphenyl)-4-(4-(hydroxydiphenylm...)

Kd: 302nMAssay Description:Inhibition of specific binding of [3H]mepyramine to Histamine 1 receptors in guinea-pigMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM22879((1R)-1-(4-tert-butylphenyl)-4-[4-(hydroxydiphenylm...)

Kd: 380nMAssay Description:Inhibition of specific binding of [3H]mepyramine to Histamine 1 receptors in guinea-pigMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM86737(UR-AK22)

Kd: 562nMAssay Description:Antagonist activity at histamine H1 receptor in guinea pig ileum assessed as inhibition of histamine-induced positive chronotropic activityMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM86735(UR-AK26)

Kd: 575nMAssay Description:Antagonist activity at histamine H1 receptor in guinea pig ileum assessed as inhibition of histamine-induced positive chronotropic activityMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50275884(CHEMBL471413 | N1-(3,3-Diphenylpropanoyl)-N2-[3-(1...)

Kd: 741nMAssay Description:Antagonist activity at histamine H1 receptor in guinea pig ileum assessed as inhibition of histamine-induced positive chronotropic activityMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM86742(UR-AK64)

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50411494(CHEMBL429458)

Kd: >1.00E+3nMAssay Description:Antagonist activity at histamine H1 receptor in guinea pig ileum assessed as inhibition of histamine-induced longitudinal smooth muscle contractionMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50228551(4-(4-fluoro-benzoyl)-1-[4-(3-piperidin-1-yl-propox...)

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50377986(CHEMBL483406 | UR-AK24)

Kd: 1.35E+3nMAssay Description:Antagonist activity at histamine H1 receptor in guinea pig ileum assessed as inhibition of histamine-induced positive chronotropic activityMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM22566(5-chloro-2-[(4-methylpiperazin-1-yl)carbonyl]-1H-i...)

Kd: 1.58E+3nMAssay Description:Antagonist activity at H1R in guinea pig ileum assessed as inhibition of histamine-induced muscle contraction after 15 minsMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM86747(UR-AK67)

Kd: 1.82E+3nMAssay Description:Antagonist activity at histamine H1 receptor in guinea pig ileum assessed as inhibition of histamine-induced positive chronotropic activityMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50118160((1-Cyclopropyl-ethyl)-carbamic acid 3-(1H-imidazol...)

Kd: 2.00E+3nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM86745(UR-AK51)

Kd: 2.14E+3nMAssay Description:Antagonist activity at histamine H1 receptor in guinea pig ileum assessed as inhibition of histamine-induced positive chronotropic activityMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM86740(UR-AK24 | UR-AK57)

Kd: 2.19E+3nMAssay Description:Antagonist activity at histamine H1 receptor in guinea pig ileum assessed as inhibition of histamine-induced positive chronotropic activityMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM86741(UR-AK59)

Kd: 2.34E+3nMAssay Description:Antagonist activity at histamine H1 receptor in guinea pig ileum assessed as inhibition of histamine-induced positive chronotropic activityMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM86744(UR-AK62)

Kd: 2.45E+3nMAssay Description:Antagonist activity at histamine H1 receptor in guinea pig ileum assessed as inhibition of histamine-induced positive chronotropic activityMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50343846(3-(1H-Imidazol-4-yl)propyl2-cyclohexylbutylcarbama...)

Kd: >3.02E+3nMAssay Description:Antagonist activity at histamine H1 receptor in guinea-pig ileumMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM22884(2-[3-(1H-imidazol-5-yl)propyl]-1-(2-{[(5-methyl-1H...)

Kd: 3.39E+3nMAssay Description:Antagonist activity at histamine H1 receptor in guinea pig ileum assessed as inhibition of histamine-induced positive chronotropic activityMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50126899(1-[4-(4-Piperidin-1-ylmethyl-benzyloxy)-phenyl]-et...)

Kd: 3.47E+3nMAssay Description:Potency at histamine H1 receptor subtype, was tested on guinea pig right ileumMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50413171(CHEMBL472273)

Kd: 3.72E+3nMAssay Description:Antagonist activity at histamine H1 receptor in guinea pig ileum assessed as inhibition of histamine-induced positive chronotropic activityMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50413173(CHEMBL513056)

Kd: 4.27E+3nMAssay Description:Antagonist activity at histamine H1 receptor in guinea pig ileum assessed as inhibition of histamine-induced positive chronotropic activityMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50126884(1-[4-(4-Piperidin-1-ylmethyl-benzyloxy)-phenyl]-et...)

Kd: 4.57E+3nMAssay Description:Potency at histamine H1 receptor subtype, was tested on guinea pig right ileumMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50413174(CHEMBL513755)

Kd: 4.68E+3nMAssay Description:Antagonist activity at histamine H1 receptor in guinea pig ileum assessed as inhibition of histamine-induced positive chronotropic activityMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50275983(CHEMBL472441 | N1-[3-(1H-Imidazol-4-yl)propyl]-N2-...)

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM86738(UR-AK46)

Kd: 5.13E+3nMAssay Description:Antagonist activity at histamine H1 receptor in guinea pig ileum assessed as inhibition of histamine-induced positive chronotropic activityMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM86743(UR-AK49)

Kd: 6.17E+3nMAssay Description:Antagonist activity at histamine H1 receptor in guinea pig ileum assessed as inhibition of histamine-induced positive chronotropic activityMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50126895(1-[4-(4-Piperidin-1-ylmethyl-benzyloxy)-phenyl]-et...)

Kd: 7.94E+3nMAssay Description:Potency at histamine H1 receptor subtype, was tested on guinea pig right ileumMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50118153((Cyclohexyl-phenyl-methyl)-carbamic acid 3-(1H-imi...)

Kd: 7.94E+3nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50126902(1-[4-(4-Pyrrolidin-1-ylmethyl-benzyloxy)-phenyl]-e...)

Kd: 9.33E+3nMAssay Description:Potency at histamine H1 receptor subtype, was tested on guinea pig right ileumMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50413181(CHEMBL499301)

Kd: 9.77E+3nMAssay Description:Antagonist activity at histamine H1 receptor in guinea pig ileum assessed as inhibition of histamine-induced positive chronotropic activityMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50118152(4-[3-(5,5-Dimethyl-hexyloxy)-propyl]-1H-imidazole;...)

Kd: 1.00E+4nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM86736(UR-AK68)

Kd: >1.00E+4nMAssay Description:Antagonist activity at histamine H1 receptor in guinea pig ileum assessed as inhibition of histamine-induced positive chronotropic activityMore data for this Ligand-Target Pair

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Histamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Regensburg

Curated by ChEMBL

BDBM50343847(3-(1H-Imidazol-4-yl)propyl2-cyclohexylpropylcarbam...)

Kd: 1.07E+4nMAssay Description:Antagonist activity at histamine H1 receptor in guinea-pig ileumMore data for this Ligand-Target Pair

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