Affinity DataIC50: 0.0100nMAssay Description:In vitro inhibition of estrogen-stimulated MCF-7 cell proliferationMore data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataIC50: 0.0460nMAssay Description:Antagonist activity at ERbeta (unknown origin) by cell-based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of 17-beta-estradiol (10e-11 M) mediated MCF-7 cell proliferationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.140nMAssay Description:Inhibition of estradiol-stimulated T-47D cell proliferation.More data for this Ligand-Target Pair
Affinity DataIC50: 0.140nMAssay Description:Inhibition of estradiol-stimulated T-47D cell proliferation.More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Antagonist effect in breast tissue was assayed by inhibition of estrogen stimulated MCF-7 cell proliferationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of estradiol-stimulated MCF-7 breast adenocarcinoma cell proliferationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:In vitro inhibition of estrogen-stimulated MCF-7 cell proliferationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Antagonism of estrogen action in a mammary tumor cell line was assayed via inhibition of MCF-7 cell proliferation stimulated by 10 e-11 M 17-beta-est...More data for this Ligand-Target Pair
Affinity DataIC50: 0.210nMAssay Description:Inhibition of ER-MDA-MB 231 breast cancer cell proliferation over 200 hrMore data for this Ligand-Target Pair
Affinity DataIC50: 0.220nMAssay Description:Inhibition of ER-MDA-MB 231 breast cancer cell proliferation over 200 hrMore data for this Ligand-Target Pair
Affinity DataIC50: 0.243nMAssay Description:Inhibition of estradiol-stimulated T-47D cell proliferation.More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Binding affinity to human ERbetaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Binding affinity to human ERbetaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Antagonist activity at ERbeta expressed in HEK293/Gal4 cells incubated for 24 hrs in presence of di-arylpropionitrile by luciferase reporter gene ass...More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Displacement of fluorescent labeled 17beta-estradiol from human ERbeta ligand binding domain by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Antagonism of estrogen action in a mammary tumor cell line was assayed via inhibition of MCF-7 cell proliferation stimulated by 10 e-11 M 17-beta-est...More data for this Ligand-Target Pair
Affinity DataIC50: 0.340nMAssay Description:Inhibition of 17-beta-estradiol (10e-11 M) mediated MCF-7 cell proliferationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.350nMAssay Description:Binding affinity for human Estrogen receptor betaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibition of [3H]-17-beta-estradiol binding to human estrogen receptor beta expressed in Escherichia coliMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Binding affinity for human Estrogen receptor betaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Displacement of [3H]17-beta-estradiol from Estrogen receptor of rabbit uterine tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Antagonism of estrogen action in a mammary tumor cell line was assayed via inhibition of MCF-7 cell proliferation stimulated by 10 e-11 M 17-beta-est...More data for this Ligand-Target Pair
Affinity DataIC50: 0.520nMAssay Description:Inhibition of 17-beta-estradiol (10e-11 M) mediated MCF-7 cell proliferationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.550nMAssay Description:Inhibition of estradiol-stimulated ZR-75-1-cell proliferationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.550nMAssay Description:Displacement of fluorescein-labeled estradiol (fluoromone) from human recombinant full-length estrogen receptor beta after 2 hrs by fluorescence pola...More data for this Ligand-Target Pair
Affinity DataIC50: 0.579nMAssay Description:Agonist activity at GAL4 DNA-binding domain fused ERbeta (unknown origin) ligand binding domain expressed in UAS-bla GripTite 293 cells assessed as b...More data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibition of binding to recombinant human ERbeta by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.631nMAssay Description:Antagonist activity at ER-beta (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.640nMAssay Description:Inhibition of fluormone ES2 binding to estrogen receptor beta after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.670nMAssay Description:Displacement of [3H]17-beta estradiol from GST-fused human recombinant ERbeta ligand binding domain expressed in Escherichia coli BL21alpha cells inc...More data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Antagonist effect against 10 pM 17-beta-estradiol induced MCF-7 cell proliferationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Inhibitory activity against Estrogen receptor by displacement of [3H]17-beta-estradiol in ER-rich cytosol from rabbit uterine tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Displacement of fluorescein labeled estradiol from human recombinant ERbeta expressed in baculovirus infected insect cells by fluorescence polarizati...More data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Antagonism of estrogen action in a mammary tumor cell line was assayed via inhibition of MCF-7 cell proliferation stimulated by 10 e-11 M 17-beta-est...More data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Binding affinity for estrogen receptor of rabbit uterine skeletal muscle tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 0.75nMAssay Description:Inhibition of ER-MDA-MB 231 breast cancer cell proliferation over 200 hrMore data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Antagonism of estrogen action in a mammary tumor cell line was assayed via inhibition of MCF-7 cell proliferation stimulated by 10 e-11 M 17-beta-est...More data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Binding affinity to human ERbetaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Antagonism of estrogen action in a mammary tumor cell line was assayed via inhibition of MCF-7 cell proliferation stimulated by 10 e-11 M 17-beta-est...More data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Antagonist effect in breast tissue was assayed by inhibition of estrogen stimulated MCF-7 cell proliferationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.820nMAssay Description:Displacement of fluorescent-labeled E2 from LBD of ERbeta (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.890nMAssay Description:Antagonist activity at ERbeta (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Antagonist effect against 10 pM 17-beta-estradiol induced MCF-7 cell proliferationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Inhibition of binding to recombinant human ERbeta by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Binding affinity to human ERbetaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Inhibitory activity against Estrogen receptor by displacement of [3H]17-beta-estradiol in ER-rich cytosol from rabbit uterine tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:In vitro inhibition of estrogen-stimulated MCF-7 cell proliferationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Inhibitory activity against Estrogen receptor by displacement of [3H]17-beta-estradiol in ER-rich cytosol from rabbit uterine tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 0.940nMAssay Description:Displacement of fluorescein-labeled estradiol (fluoromone) from human recombinant full-length estrogen receptor beta after 2 hrs by fluorescence pola...More data for this Ligand-Target Pair
