Compile Data Set for Download or QSAR
maximum 50k data
Found 29 of kd for UniProtKB: P04637
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50404458(CHEMBL4162051)
Affinity DataKd:  4.00E+3nMAssay Description:Binding affinity to N-terminal His6-tagged p53 DNA binding domain Y220C mutant (94 to 312 residues) (unknown origin) expressed in Escherichia coli C4...More data for this Ligand-Target Pair
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50404096(CHEMBL4170894)
Affinity DataKd:  1.00E+4nMAssay Description:Binding affinity to p53 Y220C mutant (unknown origin)More data for this Ligand-Target Pair
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50404081(CHEMBL4168439)
Affinity DataKd:  1.40E+4nMAssay Description:Binding affinity to N-terminal His6-tagged p53 DNA binding domain Y220C mutant (94 to 312 residues) (unknown origin) expressed in Escherichia coli C4...More data for this Ligand-Target Pair
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50404078(CHEMBL4172014)
Affinity DataKd:  2.00E+4nMAssay Description:Binding affinity to 15N-labeled T-p53 DNA binding domain Y220C mutant (94 to 312 residues) (unknown origin) expressed in Escherichia coli C41 by HSQC...More data for this Ligand-Target Pair
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50404079(CHEMBL4165245)
Affinity DataKd:  2.10E+4nMAssay Description:Binding affinity to N-terminal His6-tagged p53 DNA binding domain Y220C mutant (94 to 312 residues) (unknown origin) expressed in Escherichia coli C4...More data for this Ligand-Target Pair
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50404079(CHEMBL4165245)
Affinity DataKd:  2.10E+4nMAssay Description:Binding affinity to p53 Y220C mutant (unknown origin)More data for this Ligand-Target Pair
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50404092(CHEMBL4168045)
Affinity DataKd:  2.20E+4nMAssay Description:Binding affinity to N-terminal His6-tagged p53 DNA binding domain Y220C mutant (94 to 312 residues) (unknown origin) expressed in Escherichia coli C4...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50403663(CHEMBL4164612)
Affinity DataKd:  3.00E+4nMAssay Description:Binding affinity to 15N-labeled T-p53 DNA binding domain Y220C mutant (94 to 312 residues) (unknown origin) expressed in Escherichia coli C41 by HSQC...More data for this Ligand-Target Pair
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50404082(CHEMBL4176302)
Affinity DataKd:  3.00E+4nMAssay Description:Binding affinity to N-terminal His6-tagged p53 DNA binding domain Y220C mutant (94 to 312 residues) (unknown origin) expressed in Escherichia coli C4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50403663(CHEMBL4164612)
Affinity DataKd:  3.00E+4nMAssay Description:Binding affinity to N-terminal His6-tagged p53 DNA binding domain Y220C mutant (94 to 312 residues) (unknown origin) expressed in Escherichia coli C4...More data for this Ligand-Target Pair
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50403664(CHEMBL4168664)
Affinity DataKd:  3.00E+4nMAssay Description:Binding affinity to N-terminal His6-tagged p53 DNA binding domain Y220C mutant (94 to 312 residues) (unknown origin) expressed in Escherichia coli C4...More data for this Ligand-Target Pair
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50404088(CHEMBL4160123)
Affinity DataKd:  3.30E+4nMAssay Description:Binding affinity to N-terminal His6-tagged p53 DNA binding domain Y220C mutant (94 to 312 residues) (unknown origin) expressed in Escherichia coli C4...More data for this Ligand-Target Pair
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50404457(CHEMBL4164831)
Affinity DataKd:  5.00E+4nMAssay Description:Binding affinity to N-terminal His6-tagged p53 DNA binding domain Y220C mutant (94 to 312 residues) (unknown origin) expressed in Escherichia coli C4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50404068(CHEMBL4175464)
Affinity DataKd:  6.00E+4nMAssay Description:Binding affinity to N-terminal His6-tagged p53 DNA binding domain Y220C mutant (94 to 312 residues) (unknown origin) expressed in Escherichia coli C4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50404093(CHEMBL4163490)
Affinity DataKd:  6.30E+4nMAssay Description:Binding affinity to N-terminal His6-tagged p53 DNA binding domain Y220C mutant (94 to 312 residues) (unknown origin) expressed in Escherichia coli C4...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50404075(CHEMBL4176523)
Affinity DataKd:  7.00E+4nMAssay Description:Binding affinity to N-terminal His6-tagged p53 DNA binding domain Y220C mutant (94 to 312 residues) (unknown origin) expressed in Escherichia coli C4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50485898(CHEMBL2180125)
Affinity DataKd:  1.05E+5nMAssay Description:Binding affinity to p53 Y220C mutant by NMR spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50404087(CHEMBL4175243)
Affinity DataKd:  1.08E+5nMAssay Description:Binding affinity to N-terminal His6-tagged p53 DNA binding domain Y220C mutant (94 to 312 residues) (unknown origin) expressed in Escherichia coli C4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50404456(CHEMBL4168268)
Affinity DataKd:  1.13E+5nMAssay Description:Binding affinity to N-terminal His6-tagged p53 DNA binding domain Y220C mutant (94 to 312 residues) (unknown origin) expressed in Escherichia coli C4...More data for this Ligand-Target Pair
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50404083(CHEMBL4171798)
Affinity DataKd:  1.16E+5nMAssay Description:Binding affinity to N-terminal His6-tagged p53 DNA binding domain Y220C mutant (94 to 312 residues) (unknown origin) expressed in Escherichia coli C4...More data for this Ligand-Target Pair
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50404095(CHEMBL4171387)
Affinity DataKd:  1.22E+5nMAssay Description:Binding affinity to N-terminal His6-tagged p53 DNA binding domain Y220C mutant (94 to 312 residues) (unknown origin) expressed in Escherichia coli C4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50404069(CHEMBL4161418)
Affinity DataKd:  1.39E+5nMAssay Description:Binding affinity to N-terminal His6-tagged p53 DNA binding domain Y220C mutant (94 to 312 residues) (unknown origin) expressed in Escherichia coli C4...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50403665(CHEMBL1235116)
Affinity DataKd:  1.40E+5nMAssay Description:Binding affinity to p53 Y220C mutant (unknown origin)More data for this Ligand-Target Pair
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50403665(CHEMBL1235116)
Affinity DataKd:  1.40E+5nMAssay Description:Binding affinity to p53 Y220C mutant by NMR spectroscopyMore data for this Ligand-Target Pair
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50485897(CHEMBL1390581)
Affinity DataKd:  2.13E+5nMAssay Description:Binding affinity to p53 Y220C mutant by NMR spectroscopyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50403666(CHEMBL4160358)
Affinity DataKd:  3.06E+5nMAssay Description:Binding affinity to N-terminal His6-tagged p53 DNA binding domain Y220C mutant (94 to 312 residues) (unknown origin) expressed in Escherichia coli C4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50404084(CHEMBL4161192)
Affinity DataKd:  7.26E+5nMAssay Description:Binding affinity to N-terminal His6-tagged p53 DNA binding domain Y220C mutant (94 to 312 residues) (unknown origin) expressed in Escherichia coli C4...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50404080(CHEMBL1232243)
Affinity DataKd:  8.20E+5nMAssay Description:Binding affinity to p53 Y220C mutant (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCellular tumor antigen p53(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50590178(CHEMBL5183297)
Affinity DataKd: >1.00E+6nMAssay Description:Binding affinity to human T-p53C-Y220C mutant expressed in Escherichia coli BL21 pLysS by isothermal titration calorimetryMore data for this Ligand-Target Pair