BindingDB PrimarySearch

Found 533 of ic50 for UniProtKB: Q15139

O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)

IC50: 0.0800nMAssay Description:Inhibition Protein kinase C (PKC)More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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3D Structure (crystal)

O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519062(CHEMBL4442196)

IC50: 0.0900nMAssay Description:Agonist activity at Protein kinase C in human MT4 cells infected with HIV-1 NL4-3 assessed as inhibition of viral replication measured on day 3 post-...More data for this Ligand-Target Pair

PC cid PC sid

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O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519087(CHEMBL3741746)

IC50: 0.130nMAssay Description:Agonist activity at Protein kinase C in human MT4 cells infected with HIV-1 NL4-3 assessed as inhibition of viral replication measured on day 3 post-...More data for this Ligand-Target Pair

PC cid PC sid

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O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519068(CHEMBL4575056)

IC50: 0.140nMAssay Description:Agonist activity at Protein kinase C in human MT4 cells infected with HIV-1 NL4-3 assessed as inhibition of viral replication measured on day 3 post-...More data for this Ligand-Target Pair

PC cid PC sid

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O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519060(CHEMBL4528495)

IC50: 0.150nMAssay Description:Agonist activity at Protein kinase C in human MT4 cells infected with HIV-1 NL4-3 assessed as inhibition of viral replication measured on day 3 post-...More data for this Ligand-Target Pair

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O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519083(CHEMBL4538431)

IC50: 0.170nMAssay Description:Agonist activity at Protein kinase C in human MT4 cells infected with HIV-1 NL4-3 assessed as inhibition of viral replication measured on day 3 post-...More data for this Ligand-Target Pair

PC cid PC sid

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O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519084(CHEMBL4443190)

IC50: 0.180nMAssay Description:Agonist activity at Protein kinase C in human MT4 cells infected with HIV-1 NL4-3 assessed as inhibition of viral replication measured on day 3 post-...More data for this Ligand-Target Pair

PC cid PC sid

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O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519069(CHEMBL4435580)

IC50: 0.220nMAssay Description:Agonist activity at Protein kinase C in human MT4 cells infected with HIV-1 NL4-3 assessed as inhibition of viral replication measured on day 3 post-...More data for this Ligand-Target Pair

PC cid PC sid

Details Article PubMed

O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519063(CHEMBL4587471)

IC50: 0.360nMAssay Description:Agonist activity at Protein kinase C in human MT4 cells infected with HIV-1 NL4-3 assessed as inhibition of viral replication measured on day 3 post-...More data for this Ligand-Target Pair

PC cid PC sid

Details Article PubMed

Serine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL

BDBM50324297(4-(1-Piperazin-1-yl[2,6]naphthyridin-3-yl)pyridin-...)

IC50: 0.400nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair

NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)

IC50: 0.600nMAssay Description:Inhibition of protein kinase CMore data for this Ligand-Target Pair

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3D Structure (crystal)

Serine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL

BDBM50324315(CHEMBL1214998 | Cyclohexyl-[4-(1-piperazin-1-yl[2,...)

IC50: 0.600nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair

NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Serine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL

BDBM50324315(CHEMBL1214998 | Cyclohexyl-[4-(1-piperazin-1-yl[2,...)

IC50: 0.600nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair

NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Serine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL

BDBM50324322(4-(2-cyclohexylaminopyridin-4-yl)-6-(piperazin-1-y...)

IC50: 1nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair

NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Details Article PubMed

Serine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL

BDBM50324346(CHEMBL1215151 | Cyclohexyl-[6-piperazin-1-yl-4-(1H...)

IC50: <1nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair

NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

CHEMBL PC cid PC sid Patents Similars

Details Article PubMed

O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519064(CHEMBL4586553)

IC50: >1nMAssay Description:Agonist activity at Protein kinase C in human MT4 cells infected with HIV-1 NL4-3 assessed as inhibition of viral replication measured on day 3 post-...More data for this Ligand-Target Pair

PC cid PC sid

Details Article PubMed

O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519065(CHEMBL4578026)

PC cid PC sid

Details Article PubMed

O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519066(CHEMBL4460926)

PC cid PC sid

Details Article PubMed

O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519067(CHEMBL4443186)

PC cid PC sid

Details Article PubMed

O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519070(CHEMBL4580586)

PC cid PC sid

Details Article PubMed

O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519071(CHEMBL4585270)

PC cid PC sid

Details Article PubMed

O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519072(CHEMBL4580556)

PC cid PC sid

Details Article PubMed

O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519073(CHEMBL4536366)

PC cid PC sid

Details Article PubMed

O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519074(CHEMBL4442856)

KEGG PC cid PC sid

Details Article PubMed

O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519075(CHEMBL4558004)

PC cid PC sid

Details Article PubMed

O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519076(CHEMBL4570883)

PC cid PC sid

Details Article PubMed

O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519077(CHEMBL4470135)

PC cid PC sid

Details Article PubMed

O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519078(CHEMBL4587134)

PC cid PC sid

Details Article PubMed

O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519079(CHEMBL4451784)

PC cid PC sid

Details Article PubMed

O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519080(CHEMBL4562111)

PC cid PC sid

Details Article PubMed

O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519081(CHEMBL4537465)

PC cid PC sid

Details Article PubMed

O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519082(CHEMBL4527508)

PC cid PC sid

Details Article PubMed

O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519085(CHEMBL4444766)

PC cid PC sid

Details Article PubMed

O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519086(CHEMBL4460901)

PC cid PC sid

Details Article PubMed

O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519088(CHEMBL4475196)

PC cid PC sid

Details Article PubMed

O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519089(CHEMBL4560772)

PC cid PC sid

Details Article PubMed

O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL

BDBM50519061(CHEMBL4533733)

KEGG PC cid PC sid

Details Article PubMed

Serine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL

BDBM50324306(1-[3-(2-Cyclohexylaminopyridin-4-yl)[2,6]naphthyri...)

IC50: 1nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair

NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Serine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL

BDBM50324305(CHEMBL1214711 | N-(2-(pyrrolidin-1-yl)ethyl)-1-(3-...)

IC50: 1nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair

NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Serine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL

BDBM50324296(1-[3-(2-Cyclohexylaminopyridin-4-yl)[2,6]naphthyri...)

IC50: 1nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair

NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Serine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL

BDBM50324298(CHEMBL1215712 | {4-[1-(4-Isobutylpiperazin-1-yl)[2...)

IC50: 1nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair

NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Serine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL

BDBM50324314(1-{3-[2-(Tetrahydropyran-4-ylamino)pyridin-4-yl][2...)

IC50: 1nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair

NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Serine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL

BDBM50324325(6-Piperazin-1-yl-2'-(tetrahydropyran-4-ylamino)[2,...)

IC50: 1nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair

NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Serine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL

BDBM50324326(4'-tert-Butylcarbamoyl-2''-isopropylamino-3,4,5,6-...)

IC50: 1nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair

NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Serine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL

BDBM50324324(2'-Phenylamino-6-piperazin-1-yl[2,4']bipyridinyl-4...)

IC50: 1nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair

NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Serine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL

BDBM50324327(2'-(1-Methyl-1H-pyrazol-3-ylamino)-6-piperazin-1-y...)

IC50: 1nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair

NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Serine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL

BDBM50324328(2'-(2-Chlorophenylamino)-6-piperazin-1-yl[2,4']bip...)

IC50: 1nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair

NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Serine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL

BDBM50324323(2'-Cyclohexylamino-6-piperazin-1-yl[2,4']bipyridin...)

IC50: 1nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair

NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Serine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL

BDBM50324348(6-(piperazin-1-yl)-4-(4H-pyrazol-4-yl)-N-(tetrahyd...)

IC50: <1nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair

NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

CHEMBL PC cid PC sid Patents Similars

Details Article PubMed

Serine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL

BDBM50324347(CHEMBL1215153 | Isopropyl-[6-piperazin-1-yl-4-(1H-...)

IC50: <1nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair

NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

CHEMBL PC cid PC sid Patents Similars

Details Article PubMed

Displayed 1 to 50 (of 533 total ) | Next | Last >>

Filter my 533 hits

Targets 3▿
- O94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139 297
- Serine/threonine-protein kinase D1 234
- Protein kinase C alpha/beta/gamma/delta/epsilon/eta/theta type/Serine/threonine-protein kinase D1/D3 2
Publications 50▿
- J Med Chem 53: 5400-21 (2010) 72
- Bioorg Med Chem Lett 13: 2419-22 (2003) 32
- J Med Chem 53: 5422-38 (2010) 30
- PubChem Bioassay (2008) 30
- J Med Chem 62: 6958-6971 (2019) 30
- Bioorg Med Chem Lett 21: 1447-51 (2011) 27
- Bioorg Med Chem Lett 10: 419-22 (2000) 22
- Bioorg Med Chem Lett 9: 3307-12 (2000) 19
- PubChem Bioassay (2008) 18
- ACS Med Chem Lett 2: 154-159 (2012) 16
- J Med Chem 34: 73-8 (1991) 12
- J Med Chem 33: 1812-8 (1990) 11
- Eur J Med Chem 205: (2020) 9
- J Med Chem 42: 584-92 (1999) 9
- BMC Chem Biol 10: 5 (2010) 6
- J Nat Prod 80: 3060-3079 (2017) 5
- Bioorg Med Chem Lett 13: 3465-70 (2003) 4
- J Biol Chem 283: 33516-26 (2008) 4
- J Med Chem 41: 1631-40 (1998) 4
- J Med Chem 62: 7264-7288 (2019) 4
- Bioorg Med Chem Lett 12: 1129-32 (2002) 4
- Bioorg Med Chem Lett 11: 1993-5 (2001) 4
- Bioorg Med Chem Lett 9: 3351-6 (2000) 4
- Bioorg Med Chem Lett 7: 2415-20 (1997) 3
- Biochem J 408: 297-315 (2007) 3
- J Med Chem 61: 5881-5899 (2018) 2
- Bioorg Med Chem Lett 21: 1084-8 (2011) 2
- J Med Chem 46: 1478-83 (2003) 2
- Bioorg Med Chem Lett 21: 7155-65 (2011) 2
- Bioorg Med Chem Lett 10: 2167-70 (2001) 2
- Bioorg Med Chem Lett 13: 3835-9 (2003) 2
- Bioorg Med Chem Lett 12: 2829-31 (2002) 2
- J Med Chem 47: 4517-29 (2004) 1
- Bioorg Med Chem Lett 16: 3706-12 (2006) 1
- Eur J Med Chem 161: 456-467 (2019) 1
- Bioorg Med Chem Lett 12: 1683-6 (2002) 1
- J Med Chem 50: 3143-7 (2007) 1
- Bioorg Med Chem Lett 7: 2935-2940 (1997) 1
- Eur J Med Chem 46: 1827-34 (2011) 1
- Bioorg Med Chem Lett 16: 5122-6 (2006) 1
- Proc Natl Acad Sci U S A 104: 19936-41 (2007) 1
- J Med Chem 45: 3772-93 (2002) 1
- Bioorg Med Chem Lett 28: 2616-2621 (2018) 1
- J Med Chem 60: 8631-8646 (2017) 1
- Bioorg Med Chem 24: 521-44 (2016) 1
- Bioorg Med Chem 26: 1740-1750 (2018) 1
- Nat Chem Biol 10: 853-860 (2014) 1
- J Med Chem 62: 10691-10710 (2019) 1
- Bioorg Med Chem Lett 10: 1037-41 (2000) 1
- US Patent US9365572 (2016) 1
- ...
Institutions 38▿
- Novartis Institutes For Biomedical Research 129
- University Of Pittsburgh 74
- Millennium Pharmaceuticals 33
- Toho University 30
- Banyu Tsukuba Research Institute 22
- Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories 20
- Universit£ 13
- Ura Cnrs 1309 12
- University Of North Carolina 11
- Ku Leuven 9
- Northwestern University 6
- University Of Auckland 5
- Institute Of Molecular And Cell Biology 4
- Glaxosmithkline 4
- Celltech Therapeutics 4
- Chinese Academy Of Sciences 4
- University Of Dundee 3
- Parke-Davis Pharmaceutical Research 3
- TBA 2
- Eli Lilly 2
- Basf Bioresearch 2
- University Of Colorado 2
- Bristol-Myers Squibb Pharmaceutical Research Institute 2
- Ansaris 2
- Cephalon 2
- Msd 2
- Vertex Pharmaceuticals 1
- George Washington University 1
- University Of Florida 1
- Ewha Womans University 1
- Beijing Normal University 1
- Abbott Bioresearch Center 1
- Harvard Medical School 1
- University Of Milan 1
- Icahn School Of Medicine At Mount Sinai 1
- Xuanzhu Pharma 1
- Dongguk University 1
- Mitotix 1
- ...
Affinity: 0.080 to 3.0E+5 nM▿
- IC50 533
- Affinity ≤ nM
Xtal structures: 2
Docked structures: 0
Catalog Cmpds: 99