Compile Data Set for Download or QSAR
maximum 50k data
Found 945 of ki for UniProtKB: P08483
TargetMuscarinic acetylcholine receptor M3(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50021919(CHEMBL3298595)
Affinity DataKi:  0.0200nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M3 receptor in submandibular glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50011851(2,2-Diphenyl-propionic acid 6-methyl-6-aza-bicyclo...)
Affinity DataKi:  0.0300nMAssay Description:Inhibition of [3H]QNB binding against muscarinic acetylcholine receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50021928(CHEMBL3298599)
Affinity DataKi:  0.0490nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M3 receptor in submandibular glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50473051(CHEMBL142136)
Affinity DataKi:  0.0500nMAssay Description:In vitro for binding affinity for muscarinic acetylcholine receptors in homogenized rat brain in the presence of [3H]scopolamine.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50021904(CHEMBL3298588)
Affinity DataKi:  0.0560nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M3 receptor in submandibular glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50021922(CHEMBL3298596)
Affinity DataKi:  0.0640nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M3 receptor in submandibular glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50128836(CHEMBL143228)
Affinity DataKi:  0.0700nMAssay Description:In vitro for binding affinity for muscarinic acetylcholine receptors in homogenized rat brain in the presence of [3H]scopolamine.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50452855(Isoptpo Hyoscine | Scopolamine)
Affinity DataKi:  0.0800nMAssay Description:Inhibition of [3H]pirenzepine binding to muscarinic receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails
TargetMuscarinic acetylcholine receptor M3(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50011851(2,2-Diphenyl-propionic acid 6-methyl-6-aza-bicyclo...)
Affinity DataKi:  0.0986nMAssay Description:The compound was tested for binding activity against muscarinic acetylcholine receptor M3, using [3H]-QNB as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50021935(CHEMBL3298600)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M3 receptor in submandibular glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50011851(2,2-Diphenyl-propionic acid 6-methyl-6-aza-bicyclo...)
Affinity DataKi:  0.118nMAssay Description:Inhibition of [3H]pirenzepine binding against muscarinic acetylcholine receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50403547(ATROPEN | ATROPINE)
Affinity DataKi:  0.120nMAssay Description:Ability to displace [3H]N-methylscopolamine (NMS) from M3 receptor in rat submaxillary gland homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50021893(CHEMBL3298333)
Affinity DataKi:  0.120nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M3 receptor in submandibular glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50021938(CHEMBL3298763)
Affinity DataKi:  0.120nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M3 receptor in submandibular glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50344285(CHEMBL1779047 | quinuclidin-4-yl biphenyl-2-ylcarb...)
Affinity DataKi:  0.140nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M3 receptor in submandibular glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50450592(CHEMBL558910)
Affinity DataKi:  0.160nMAssay Description:Ability to displace [3H]N-methylscopolamine (NMS) from M3 receptor in rat submaxillary gland homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50473042(CHEMBL141269)
Affinity DataKi:  0.160nMAssay Description:In vitro for binding affinity for muscarinic acetylcholine receptors in homogenized rat brain in the presence of [3H]scopolamine.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50368152(CHEMBL318812)
Affinity DataKi:  0.166nMAssay Description:Inhibition of [3H]pirenzepine binding against muscarinic acetylcholine receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50021892(Ipratropium Bromide)
Affinity DataKi:  0.180nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M3 receptor in submandibular glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50015720((hyoscine)3-Hydroxy-2-phenyl-propionic acid 9-meth...)
Affinity DataKi:  0.180nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50021905(CHEMBL3298589)
Affinity DataKi:  0.190nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M3 receptor in submandibular glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50011851(2,2-Diphenyl-propionic acid 6-methyl-6-aza-bicyclo...)
Affinity DataKi:  0.196nMAssay Description:Inhibition of [3H]QNB binding against muscarinic acetylcholine receptor in rat heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50368152(CHEMBL318812)
Affinity DataKi:  0.197nMAssay Description:Inhibition of [3H]pirenzepine binding against muscarinic acetylcholine receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50021909(CHEMBL3298591)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M3 receptor in submandibular glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50005363((3R,4R)3-(3-Methyl-[1,2,4]oxadiazol-5-yl)-1-aza-bi...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity against Muscarinic acetylcholine receptor using [3H]-OXO-M as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50021901(CHEMBL3298334)
Affinity DataKi:  0.210nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M3 receptor in submandibular glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50368152(CHEMBL318812)
Affinity DataKi:  0.224nMAssay Description:Inhibition of [3H]QNB binding against muscarinic acetylcholine receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50471498(CHEMBL150450)
Affinity DataKi:  0.240nMAssay Description:Binding affinity against Muscarinic acetylcholine receptors using [3H]oxotremorine-M as radioligand in rat cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50241132(3-Hydroxy-2-phenyl-propionic acid 9-methyl-3-oxa-9...)
Affinity DataKi:  0.25nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50021926(CHEMBL3298598)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M3 receptor in submandibular glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50368152(CHEMBL318812)
Affinity DataKi:  0.254nMAssay Description:Inhibition of [3H]QNB binding against muscarinic acetylcholine receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50456344(CHEMBL2112942)
Affinity DataKi:  0.270nMAssay Description:Ability to displace [3H]N-methylscopolamine (NMS) from M3 receptor in rat submaxillary gland homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50368152(CHEMBL318812)
Affinity DataKi:  0.297nMAssay Description:Inhibition of [3H]QNB binding against muscarinic acetylcholine receptor in rat heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50229368(CHEMBL77793)
Affinity DataKi:  0.300nMAssay Description:Binding affinity to muscarinic acetylcholine receptor was determined in presence of [3H]OXO-M radioligand (in vitro)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50403547(ATROPEN | ATROPINE)
Affinity DataKi:  0.300nMAssay Description:The compound was tested for inhibition of [3H]NMS binding against muscarinic acetylcholine receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50296345((1R,2R,4S,5R,7S)-7-(2-hydroxy-2,2-di-thiophen-2-yl...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M3 receptor in submandibular glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50368152(CHEMBL318812)
Affinity DataKi:  0.302nMAssay Description:Inhibition of [3H]QNB binding against muscarinic acetylcholine receptor in rat heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM86231(ATR | ATROPINE | Atropine,(-) | CAS_51-55-8 | CHEM...)
Affinity DataKi:  0.310nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50471487(CHEMBL436075)
Affinity DataKi:  0.330nMAssay Description:Binding affinity against Muscarinic acetylcholine receptors using [3H]oxotremorine-M as radioligand in rat cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50403547(ATROPEN | ATROPINE)
Affinity DataKi:  0.337nMAssay Description:Inhibition of [3H]QNB binding against muscarinic acetylcholine receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50403547(ATROPEN | ATROPINE)
Affinity DataKi:  0.337nMAssay Description:Inhibition of [3H]QNB binding to muscarinic acetylcholine receptor of rat heart membrane preparation.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50471494(CHEMBL153723)
Affinity DataKi:  0.360nMAssay Description:Binding affinity against Muscarinic acetylcholine receptors using [3H]oxotremorine-M as radioligand in rat cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50021924(CHEMBL3298597)
Affinity DataKi:  0.370nMAssay Description:Displacement of [3H]-NMS from Sprague-Dawley rat muscarinic M3 receptor in submandibular glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM82372(CAS_22254-24-6 | Ipratropium | NSC_3746)
Affinity DataKi:  0.370nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50471499(CHEMBL345774)
Affinity DataKi:  0.400nMAssay Description:Binding affinity against Muscarinic acetylcholine receptor using [3H]oxotremorine-M as radioligand in rat cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM86231(ATR | ATROPINE | Atropine,(-) | CAS_51-55-8 | CHEM...)
Affinity DataKi:  0.400nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50471859(CHEMBL334387)
Affinity DataKi:  0.400nMAssay Description:Binding affinity against Muscarinic acetylcholine receptor using [3H]-OXO-M as the radioligand.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50471485(Vedaclidine)
Affinity DataKi:  0.400nMAssay Description:Binding affinity against Muscarinic acetylcholine receptors using [3H]oxotremorine-M as radioligand in rat cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50473044(CHEMBL343764)
Affinity DataKi:  0.410nMAssay Description:In vitro for binding affinity for muscarinic acetylcholine receptors in homogenized rat brain in the presence of [3H]scopolamine.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50471492(CHEMBL150293)
Affinity DataKi:  0.420nMAssay Description:Binding affinity against Muscarinic acetylcholine receptors using [3H]oxotremorine-M as radioligand in rat cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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