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Found 65 of ic50 for UniProtKB: P00761
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50044092(spumigin E)
Affinity DataIC50: <100nMAssay Description:Inhibition of pig pancreas trypsin type IX-S using Boc-Gln-Ala-Arg-MCA substrate by 7-amino-4-methylcoumarin release based spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50286441((S)-2-((S)-2-Acetylamino-4-(S)-methyl-pentanoylami...)
Affinity DataIC50: >200nMAssay Description:Inhibition of pig pancreas trypsin type IX-SMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50044094(CHEMBL3325623)
Affinity DataIC50:  350nMAssay Description:Inhibition of pig pancreas trypsin type IX-S using Boc-Gln-Ala-Arg-MCA substrate by 7-amino-4-methylcoumarin release based spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50286441((S)-2-((S)-2-Acetylamino-4-(S)-methyl-pentanoylami...)
Affinity DataIC50:  500nMAssay Description:Inhibition of pig pancreas trypsin type IX-S using Boc-Gln-Ala-Arg-MCA substrate by 7-amino-4-methylcoumarin release based spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50041802(1,8-dihydroxy-9(10H)-anthracenone | 1,8-dihydroxy-...)
Affinity DataIC50:  1.26E+3nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM191635(US9182402, 8)
Affinity DataIC50:  1.71E+3nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM191638(US9182402, 11)
Affinity DataIC50:  2.00E+3nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50013876(CHEMBL291278 | Methyl aspartic acid | N-Methyl asp...)
Affinity DataIC50:  2.42E+3nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM191639(US9182402, 12)
Affinity DataIC50:  3.50E+3nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM123129(1-(3-nitro-phenyl)-pyrrole-2,5-dione (17) | CID236...)
Affinity DataIC50:  3.88E+3nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085340(CHEMBL448737 | N-((S)-1-Benzyl-3-chloro-2-oxo-prop...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM191630(US9182402, 3)
Affinity DataIC50:  7.63E+3nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM191637(US9182402, 10)
Affinity DataIC50:  7.72E+3nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM191633(US9182402, 6)
Affinity DataIC50:  1.02E+4nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM191634(US9182402, 7)
Affinity DataIC50:  1.31E+4nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50069104(CHEMBL1449583 | US9182402, 4)
Affinity DataIC50:  1.96E+4nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM191632(US9182402, 2)
Affinity DataIC50: >2.00E+4nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM81467(CAS_569-65-3 | CHEMBL1085765 | Meclizine | NSC_403...)
Affinity DataIC50: >2.00E+4nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM191636(US9182402, 9)
Affinity DataIC50:  2.09E+4nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085346(CHEMBL294290 | N-((S)-1-Benzyl-3-chloro-2-oxo-prop...)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085354(CHEMBL60160 | N-((S)-1-Benzyl-3-chloro-2-oxo-propy...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM191631(US9182402, 5)
Affinity DataIC50:  3.12E+4nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50007260(2,6-Di-tert-butyl-4-[1-(3,5-di-tert-butyl-4-hydrox...)
Affinity DataIC50:  3.35E+4nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085341(CHEMBL294326 | N-((S)-1-Benzyl-3-chloro-2-oxo-prop...)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085356(CHEMBL61933 | N-((S)-1-Benzyl-3-chloro-2-oxo-propy...)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085364(CHEMBL59660 | N-((S)-1-Benzyl-3-chloro-2-oxo-propy...)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50044093(CHEMBL3325624)
Affinity DataIC50:  5.50E+4nMAssay Description:Inhibition of pig pancreas trypsin type IX-S using Boc-Gln-Ala-Arg-MCA substrate by 7-amino-4-methylcoumarin release based spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085361(CHEMBL59998 | N-((S)-1-Benzyl-3-chloro-2-oxo-propy...)
Affinity DataIC50:  7.50E+4nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085343(CHEMBL64202 | N-((S)-1-Benzyl-3-chloro-2-oxo-propy...)
Affinity DataIC50:  8.50E+4nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085352(CHEMBL62222 | N-((S)-1-Benzyl-3-chloro-2-oxo-propy...)
Affinity DataIC50:  9.70E+4nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085353(CHEMBL293590 | N-((S)-1-Benzyl-3-chloro-2-oxo-prop...)
Affinity DataIC50:  1.20E+5nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50150484((Z)-9-octadecenoic acid | (Z)-Octadec-9-enoic acid...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of pig pancreatic trypsin after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50269531((9Z)-hexadec-9-enoic acid | (Z)-9-hexadecenoic aci...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of pig pancreatic trypsin after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50269530((9Z)-tetradec-9-enoic acid | CHEMBL456732 | cis-De...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of pig pancreatic trypsin after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50269532((6,9,12)-linolenic acid | (6Z,9Z,12Z)-octadeca-6,9...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of pig pancreatic trypsin after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50240347((9,12,15)-linolenic acid | (9Z,12Z,15Z)-octadeca-9...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of pig pancreatic trypsin after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM22231((9Z,12Z)-octadeca-9,12-dienoic acid | CHEMBL267476...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of pig pancreatic trypsin after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50269534((8Z,11Z,14Z)-Icosatrienoic acid | (8Z,11Z,14Z)-ico...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of pig pancreatic trypsin after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50269540(6-(8'Z,11'Z-heptadecadienyl)-salicylicacid | CHEMB...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of pig pancreatic trypsin after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085363(CHEMBL60718 | L-1-Tosylamido-2-phenylethyl chlorom...)
Affinity DataIC50:  2.00E+5nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50259930(6-(10'Z-heptadecenyl)-salicylicacid | 6-[10'(Z)-he...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of pig pancreatic trypsin after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50242188(6-(8'Z-pentadecenyl)-salicylicacid | 6-[8'(Z)-pent...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of pig pancreatic trypsin after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50242349((5Z,8Z,11Z,14Z,17Z)-5,8,11,14,17-eicosapentaenoic ...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of pig pancreatic trypsin after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM22319((5Z,8Z,11Z,14Z)-icosa-5,8,11,14-tetraenoic acid | ...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of pig pancreatic trypsin after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50269535((11Z,14Z,17Z)-Eicosa-11,14,17-trienoic acid | (11Z...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of pig pancreatic trypsin after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50269533(CHEMBL464983 | cis-11,14-eicosadienoicacid)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of pig pancreatic trypsin after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085339(((S)-1-Benzyl-3-chloro-2-oxo-propyl)-carbamic acid...)
Affinity DataIC50:  2.10E+5nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085362(CHEMBL64494 | N-((S)-1-Benzyl-3-chloro-2-oxo-propy...)
Affinity DataIC50:  2.10E+5nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085360(CHEMBL302387 | N-((S)-1-Benzyl-3-chloro-2-oxo-prop...)
Affinity DataIC50:  2.40E+5nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085348(CHEMBL60715 | N-((S)-1-Benzyl-3-chloro-2-oxo-propy...)
Affinity DataIC50:  2.60E+5nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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