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Found 8 of ic50 for UniProtKB: P06281
TargetRenin-1(Mus musculus)
Novartis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM17950((2S,4S,5S,7S)-5-amino-N-(2-carbamoyl-2,2-dimethyle...)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of mouse reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin-1(Mus musculus)
Novartis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50022867(2-[2-(2-{[7-(2-tert-Butoxycarbonylamino-3-phenyl-p...)
Affinity DataIC50:  400nMAssay Description:Inhibitory activity against mouse reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin-1(Mus musculus)
Novartis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50022862(Boc-Phe-Ala-Leu-Val-Ile-His-OMe | CHEMBL101874)
Affinity DataIC50:  500nMAssay Description:Inhibitory activity against mouse reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin-1(Mus musculus)
Novartis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50022864(Boc-Phe-(CH3)Ala-Leu-Val-Ile-His-OMe | CHEMBL31824...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory activity against mouse reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin-1(Mus musculus)
Novartis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50022866(4-[1-{3-[1-[1-(1-amino-1-methylpropylcarboxamido)-...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibitory activity against mouse reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin-1(Mus musculus)
Novartis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50022863(2-[2-(2-{[7-(2-tert-Butoxycarbonylamino-3-phenyl-p...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibitory activity against mouse reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin-1(Mus musculus)
Novartis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50022865(Boc-Phe-His-Leu-Val-Ile-His-OMe | CHEMBL321937)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibitory activity against mouse reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin-1(Mus musculus)
Novartis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50022868(2-[2-(2-{[7-(2-tert-Butoxycarbonylamino-3-phenyl-p...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against mouse reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed