Compile Data Set for Download or QSAR
maximum 50k data
Found 29 of ec50 for UniProtKB: P11416
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataEC50:  1.20nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataEC50:  1.5nMAssay Description:Transactivation of mouse Gal4-fused RARalpha-LBD expressed in COS-7 cells after 1 day by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526321(CHEMBL4572914)
Affinity DataEC50:  4nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM50048292(6-[4-Methoxy-3-(1-methyl-cyclohexyl)-phenyl]-napht...)
Affinity DataEC50:  9.20nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526312(CHEMBL4449668 | US10752616, Code No. BHBA-007)
Affinity DataEC50:  16nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526311(CHEMBL4588745)
Affinity DataEC50:  18nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526317(CHEMBL4437942)
Affinity DataEC50:  18nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM50064254((2E,4E,6E,8Z)-3,7-Dimethyl-9-(2,6,6-trimethyl-cycl...)
Affinity DataEC50:  18nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid A receptor RAR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526315(CHEMBL4439399 | US10752616, Code No. BHBA-019)
Affinity DataEC50:  19nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataEC50:  22nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid A receptor RAR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526314(CHEMBL4459692 | US10752616, Code No. BHBA-001)
Affinity DataEC50:  26nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526325(CHEMBL4438880 | US10752616, Code No. BHBA-021)
Affinity DataEC50:  30nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526322(CHEMBL4442948)
Affinity DataEC50:  31nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM50031460((2E,4E,6E)-8-[3-Ethyl-2-isopropyl-cyclohex-2-en-(E...)
Affinity DataEC50:  33nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid A receptor RAR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526318(CHEMBL4215742)
Affinity DataEC50:  46nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM50064252((2Z,4E,6E)-8-[3-Ethyl-2-isopropyl-cyclohex-2-en-(E...)
Affinity DataEC50:  51nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid A receptor RAR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526324(CHEMBL4439947)
Affinity DataEC50:  58nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526319(CHEMBL4517145)
Affinity DataEC50:  60nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526316(CHEMBL4531897)
Affinity DataEC50:  61nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM50413272(AC-261066 | CHEMBL198997)
Affinity DataEC50:  70nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526313(CHEMBL4469143 | US10752616, Code No. BHBA-006)
Affinity DataEC50:  89nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526327(CHEMBL4562084 | US10752616, Code No. BHBA-023)
Affinity DataEC50:  114nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526323(CHEMBL4539676)
Affinity DataEC50:  240nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526326(CHEMBL4590840)
Affinity DataEC50:  594nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526320(CHEMBL4448702)
Affinity DataEC50:  600nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM50064255((2E,4Z,6Z)-8-[3-Ethyl-2-isopropyl-cyclohex-2-en-(E...)
Affinity DataEC50: >1.00E+3nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid A receptor RAR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM50064250((2E,4E,6E)-8-[3,4-Dihydro-2H-naphthalen-(1E)-ylide...)
Affinity DataEC50: >2.00E+3nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid A receptor RAR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM50064251((2Z,4E,6E)-8-[3,4-Dihydro-2H-naphthalen-(1E)-ylide...)
Affinity DataEC50: >2.00E+3nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid A receptor RAR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
King'S College

Curated by ChEMBL
LigandPNGBDBM50064253((2E,4Z,6Z)-8-[3,4-Dihydro-2H-naphthalen-(1E)-ylide...)
Affinity DataEC50: >2.00E+3nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid A receptor RAR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed