Compile Data Set for Download or QSAR
maximum 50k data
Found 52 of ki data for polymerid = 50001895
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066694((S)-2-[(R)-7-(3-Chloro-9H-fluoren-9-yl)-2-hydroxy-...)
Affinity DataKi:  220nMAssay Description:Inhibition of human ACLYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066694((S)-2-[(R)-7-(3-Chloro-9H-fluoren-9-yl)-2-hydroxy-...)
Affinity DataKi:  220nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50394668(CHEMBL2163366)
Affinity DataKi:  220nMAssay Description:Inhibition of human recombinant ACLYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066677((S)-2-{(R)-8-[4-Chloro-2-(3,4-dimethyl-pyrrol-1-yl...)
Affinity DataKi:  300nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066677((S)-2-{(R)-8-[4-Chloro-2-(3,4-dimethyl-pyrrol-1-yl...)
Affinity DataKi:  300nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50394671(CHEMBL2165260)
Affinity DataKi:  340nMAssay Description:Inhibition of human recombinant ACLYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50394671(CHEMBL2165260)
Affinity DataKi:  340nMAssay Description:Inhibition of human recombinant ACLYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066673((S)-2-[(R)-7-(5-Chloro-2-phenyl-indol-1-yl)-2-hydr...)
Affinity DataKi:  370nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50394670(CHEMBL2165263)
Affinity DataKi:  370nMAssay Description:Inhibition of human recombinant ACLYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066676((2S,3R)-2-[(R)-8-(2,4-Dichloro-phenyl)-2-hydroxy-o...)
Affinity DataKi:  550nMAssay Description:Inhibition of human recombinant ACLYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066676((2S,3R)-2-[(R)-8-(2,4-Dichloro-phenyl)-2-hydroxy-o...)
Affinity DataKi:  550nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50394671(CHEMBL2165260)
Affinity DataKi:  580nMAssay Description:Inhibition of human recombinant ACLYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066688((2S,3S)-2-[(R)-8-(2,4-Dichloro-phenyl)-2-hydroxy-o...)
Affinity DataKi:  620nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50394672(CHEMBL2165259)
Affinity DataKi:  620nMAssay Description:Inhibition of human recombinant ACLYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50394677(CHEMBL2165262)
Affinity DataKi:  700nMAssay Description:Competitive inhibition of human liver ACLY using varying levels of citrate as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066682((S)-2-[(R)-7-(3-Chloro-carbazol-9-yl)-2-hydroxy-he...)
Affinity DataKi:  710nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50394669(CHEMBL2165264)
Affinity DataKi:  710nMAssay Description:Inhibition of human recombinant ACLYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066689((S)-2-[(R)-8-(5-Chloro-biphenyl-2-yl)-2-hydroxy-oc...)
Affinity DataKi:  750nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066683((S)-2-((R)-8-(2,4-dichlorophenyl)-2-hydroxyoctyl)-...)
Affinity DataKi:  770nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066683((S)-2-((R)-8-(2,4-dichlorophenyl)-2-hydroxyoctyl)-...)
Affinity DataKi:  770nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066683((S)-2-((R)-8-(2,4-dichlorophenyl)-2-hydroxyoctyl)-...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibitory activity was tested agianst human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066683((S)-2-((R)-8-(2,4-dichlorophenyl)-2-hydroxyoctyl)-...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of human ACLYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066683((S)-2-((R)-8-(2,4-dichlorophenyl)-2-hydroxyoctyl)-...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of human ATP citrate lyaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066683((S)-2-((R)-8-(2,4-dichlorophenyl)-2-hydroxyoctyl)-...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of human recombinant ACLYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066672((S)-2-[(R)-8-(2-Benzyloxy-4-chloro-phenyl)-2-hydro...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066685((S)-2-[(R)-7-(5,7-Dichloro-indol-1-yl)-2-hydroxy-h...)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066692((S)-2-((S)-8-(2,4-dichlorophenyl)-2-hydroxyoctyl)-...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066687((S)-2-[(R)-8-(5-Chloro-4'-fluoro-biphenyl-2-yl)-2-...)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066680((S)-2-[(R)-8-(5-Chloro-4'-methyl-biphenyl-2-yl)-2-...)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066686((S)-2-[(R)-7-(3-Benzyl-5-chloro-indol-1-yl)-2-hydr...)
Affinity DataKi:  2.90E+3nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066678((S)-2-[(R)-7-(6-Chloro-1,2,3,4-tetrahydro-carbazol...)
Affinity DataKi:  2.90E+3nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066693((S)-2-[(R)-8-(5-Chloro-indol-1-yl)-2-hydroxy-octyl...)
Affinity DataKi:  3.20E+3nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50394678(CHEMBL2165261)
Affinity DataKi:  3.20E+3nMAssay Description:Competitive inhibition of human liver ACLY using varying levels of citrate as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066699((S)-2-[(R)-7-(5-Chloro-indol-1-yl)-2-hydroxy-hepty...)
Affinity DataKi:  3.50E+3nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066702((S)-2-[(R)-8-(4-Chloro-2-pyrrol-1-yl-phenyl)-2-hyd...)
Affinity DataKi:  3.90E+3nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066695((S)-2-[(R)-8-(5,4'-Dichloro-biphenyl-2-yl)-2-hydro...)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066700((S)-2-[(R)-8-(5-Chloro-4'-methoxy-biphenyl-2-yl)-2...)
Affinity DataKi:  5.10E+3nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066701((R)-2-[(S)-8-(2,4-Dichloro-phenyl)-1-hydroxy-octyl...)
Affinity DataKi:  5.70E+3nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066675((S)-2-[(R)-7-(5-Chloro-3-methyl-indol-1-yl)-2-hydr...)
Affinity DataKi:  9.50E+3nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066698((S)-2-[(R)-7-(5-Chloro-3-phenyl-indol-1-yl)-2-hydr...)
Affinity DataKi:  1.10E+4nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066691((S)-2-[(R)-7-(5-Chloro-2-methyl-indol-1-yl)-2-hydr...)
Affinity DataKi:  1.30E+4nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066674((R)-2-[(S)-9-(2,4-Dichloro-phenyl)-1-hydroxy-nonyl...)
Affinity DataKi:  1.80E+4nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066703((S)-2-[(R)-8-(4-Chloro-2-methoxy-phenyl)-2-hydroxy...)
Affinity DataKi:  1.90E+4nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066681((S)-2-Hydroxy-2-[(R)-2-hydroxy-8-(5,2',4'-trichlor...)
Affinity DataKi:  2.10E+4nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50052987(2-[6-(4-Chloro-2-nitro-phenyl)-hexylsulfanylmethyl...)
Affinity DataKi:  2.60E+4nMAssay Description:Inhibitory activity against rat ATP-Citrate Lyase activity was measured by the maleate dehydrogenase catalyzed reduction of oxaloacetate by NADHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066690((S)-2-[(R)-7-(6-Chloro-indol-1-yl)-2-hydroxy-hepty...)
Affinity DataKi:  4.10E+4nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066679((S)-2-[(R)-7-(5-Chloro-3-nitro-indol-1-yl)-2-hydro...)
Affinity DataKi:  6.40E+4nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50053013(2-[6-(3,5-Dichloro-pyridin-4-yl)-hexylsulfanylmeth...)
Affinity DataKi:  1.21E+5nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase activity was measured by the maleate dehydrogenase catalyzed reduction of oxaloacetat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50066704((S)-2-[(R)-6-(5-Chloro-indol-1-yl)-2-hydroxy-hexyl...)
Affinity DataKi:  1.60E+5nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50052984(2-Hydroxy-2-(3-naphthalen-2-yl-propylsulfanylmethy...)
Affinity DataKi:  3.00E+5nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase activity was measured by the maleate dehydrogenase catalyzed reduction of oxaloacetat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 52 total ) | Next | Last >>
Jump to: