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Found 14 of ki for UniProtKB: P06935
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50513894(CHEMBL4457231)
Affinity DataKi:  120nMAssay Description:Inhibition of West Nile virus NS2B (47 residues)-NS3 (184 residues) protease expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50030459(CHEMBL3344321)
Affinity DataKi:  130nMAssay Description:Inhibition of West Nile virus NS2B-NS3 proteaseMore data for this Ligand-Target Pair
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50587014(CHEMBL5094815)
Affinity DataKi:  343nMAssay Description:Competitive inhibition of C-terminal His-tagged WNV NSB2 (52 to 96 amino acids)-NS3 (1 to 184 amino acids) protease expressed in Escherichia coli BL2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50109138(CHEMBL3601351)
Affinity DataKi:  820nMAssay Description:Inhibition of WNV NS2B-NS3 protease expressed in Escherichia coli BL21 lambda (DE3) cells using Abz-Gly-Leu-Lys-Arg-Gly-Gly-3-(NO2)Tyr as substrate p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50542823(CHEMBL4633312)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of West Nile virus NS2B-NS3 protease expressed in Escherichia coli BL21 lambda (DE3) cells using Abz-Gly-Leu-Lys-Arg-Gly-Gly-3-(NO2)Tyr as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50109138(CHEMBL3601351)
Affinity DataKi:  1.30E+3nMAssay Description:Competitive inhibition of WNV NS2B-NS3 protease expressed in Escherichia coli BL21 lambda (DE3) cells using Abz-Gly-Leu-Lys-Arg-Gly-Gly-3-(NO2)Tyr as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50030461(CHEMBL3344320)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of West Nile virus NS2B-NS3 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50513895(CHEMBL1797630)
Affinity DataKi:  4.90E+3nMAssay Description:Inhibition of West Nile virus NS2B-NS3 protease preincubated for 1 hr followed by Pyr-RTKR-AMC addition and measured after 30 mins by fluorescence me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50538478(CHEMBL4634219)
Affinity DataKi:  7.40E+3nMAssay Description:Inhibition of C-terminal His6-tagged West Nile virus NS2B (52 to 96 residues)-G4SG4-NS3 (1 to 184 residues) expressed in Escherichia coli BL21(DE3) c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50513898(CHEMBL4587076)
Affinity DataKi:  8.00E+3nMAssay Description:Inhibition of West Nile virus NS2B-NS3 protease preincubated for 10 mins followed by Np-KKR-pNA addition and measured every 5 secs for 2 mins by fluo...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50542799(CHEMBL4649655)
Affinity DataKi:  1.20E+4nMAssay Description:Inhibition of West Nile virus NS2B-NS3 protease expressed in Escherichia coli BL21 lambda (DE3) cells using Abz-Gly-Leu-Lys-Arg-Gly-Gly-3-(NO2)Tyr as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50538477(CHEMBL4633138)
Affinity DataKi:  2.55E+4nMAssay Description:Inhibition of C-terminal His6-tagged West Nile virus NS2B (52 to 96 residues)-G4SG4-NS3 (1 to 184 residues) expressed in Escherichia coli BL21(DE3) c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50026765(CHEMBL3335494)
Affinity DataKi:  4.90E+4nMAssay Description:Inhibition of West Nile virus serotype 2 NS2B-NS3 protease by homogeneous fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50026808(CHEMBL2440341)
Affinity DataKi:  9.25E+4nMAssay Description:Inhibition of West Nile virus NS2B-NS3 protease preincubated for 15 mins followed by Abz-Gly-Leu-Lys-Arg-Gly-Gly-3-(NO2)Tyr addition and measured for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed