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Found 33 of ic50 for UniProtKB: A0A140VJJ9
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50208436(CHEMBL3885040)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of recombinant GGT1 (unknown origin) using GGPP as substrate preincubated for 5 mins followed by protein addition measured over 20 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50208427(CHEMBL3884872)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of recombinant GGT1 (unknown origin) using GGPP as substrate preincubated for 5 mins followed by protein addition measured over 20 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM14713(GGTI-DU40 | N-[(1S)-1-carbamoyl-2-phenylethyl]-4-{...)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of recombinant GGT1 (unknown origin) using GGPP as substrate preincubated for 5 mins followed by protein addition measured over 20 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50208433(CHEMBL3885443)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition of recombinant GGT1 (unknown origin) using GGPP as substrate preincubated for 5 mins followed by protein addition measured over 20 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50208426(CHEMBL3883795)
Affinity DataIC50:  9.90E+3nMAssay Description:Inhibition of recombinant GGT1 (unknown origin) using GGPP as substrate preincubated for 5 mins followed by protein addition measured over 20 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50208438(CHEMBL3885188)
Affinity DataIC50:  1.16E+4nMAssay Description:Inhibition of recombinant GGT1 (unknown origin) using GGPP as substrate preincubated for 5 mins followed by protein addition measured over 20 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50248772(2-(1,3-benzodioxol-5-yl)-N,N',4-trimethyl-10Hpheno...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of gamma-glutamyltranspeptidase (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50248738(2-(2-Chlorophenyl)-N,N',4-trimethyl-10Hphenothiazi...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of gamma-glutamyltranspeptidase (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50248626(2-(2-Chlorophenyl)-N,N',4-trimethyl-2,10-dihydro-1...)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of gamma-glutamyltranspeptidase (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50208434(CHEMBL3884826)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of recombinant GGT1 (unknown origin) using GGPP as substrate preincubated for 5 mins followed by protein addition measured over 20 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50208431(CHEMBL3883522)
Affinity DataIC50:  1.97E+4nMAssay Description:Inhibition of recombinant GGT1 (unknown origin) using GGPP as substrate preincubated for 5 mins followed by protein addition measured over 20 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50248739(2-(4-Chlorophenyl)-N,N',4-trimethyl-10Hphenothiazi...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of gamma-glutamyltranspeptidase (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50248736(2-Phenyl-N,N',4-trimethyl-10H-phenothiazine-1,3-di...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of gamma-glutamyltranspeptidase (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50248624(2-Phenyl-N,N',4-trimethyl-2,10-dihydro-1Hphenothia...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of gamma-glutamyltranspeptidase (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50248771(2-(4-Methoxyphenyl)-N,N',4-trimethyl-10Hphenothiaz...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of gamma-glutamyltranspeptidase (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50248773(2-(4-Nitrophenyl)-N,N',4-trimethyl-10Hphenothiazin...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of gamma-glutamyltranspeptidase (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50248625(2-(2-Methylphenyl)-N,N',4-trimethyl-2,10-dihydro-1...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of gamma-glutamyltranspeptidase (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50208423(CHEMBL3884658)
Affinity DataIC50:  2.29E+4nMAssay Description:Inhibition of recombinant GGT1 (unknown origin) using GGPP as substrate preincubated for 5 mins followed by protein addition measured over 20 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50248701(2-(4-Methoxyphenyl)-N,N',4-trimethyl-2,10-dihydro-...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of gamma-glutamyltranspeptidase (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50248737(2-(2-Methylphenyl)-N,N',4-trimethyl-10Hphenothiazi...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of gamma-glutamyltranspeptidase (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50208437(CHEMBL3884852)
Affinity DataIC50:  2.63E+4nMAssay Description:Inhibition of recombinant GGT1 (unknown origin) using GGPP as substrate preincubated for 5 mins followed by protein addition measured over 20 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50208430(CHEMBL3884083)
Affinity DataIC50:  2.69E+4nMAssay Description:Inhibition of recombinant GGT1 (unknown origin) using GGPP as substrate preincubated for 5 mins followed by protein addition measured over 20 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50248770(2-(2-Methoxyphenyl)-N,N',4-trimethyl-10Hphenothiaz...)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of gamma-glutamyltranspeptidase (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50248702(2-(1,3-Benzodioxol-5-yl)-N,N',4-trimethyl-2,10-dih...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of gamma-glutamyltranspeptidase (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50248700(2-(2-Methoxyphenyl)-N,N',4-trimethyl-2,10-dihydro-...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of gamma-glutamyltranspeptidase (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50208429(CHEMBL3883400)
Affinity DataIC50:  3.19E+4nMAssay Description:Inhibition of recombinant GGT1 (unknown origin) using GGPP as substrate preincubated for 5 mins followed by protein addition measured over 20 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50208435(CHEMBL3885260)
Affinity DataIC50:  3.48E+4nMAssay Description:Inhibition of recombinant GGT1 (unknown origin) using GGPP as substrate preincubated for 5 mins followed by protein addition measured over 20 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50248655(2-(4-Chlorophenyl)-N,N',4-trimethyl-2,10-dihydro-1...)
Affinity DataIC50: >3.50E+4nMAssay Description:Inhibition of gamma-glutamyltranspeptidase (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM22360(2-(acetyloxy)benzoate | 2-(acetyloxy)benzoic acid ...)
Affinity DataIC50:  3.60E+4nMAssay Description:Inhibition of gamma-glutamyltranspeptidase (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50248703(2-(4-Nitrophenyl)-N,N',4-trimethyl-2,10-dihydro-1H...)
Affinity DataIC50:  3.60E+4nMAssay Description:Inhibition of gamma-glutamyltranspeptidase (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50208425(CHEMBL3884603)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant GGT1 (unknown origin) using GGPP as substrate preincubated for 5 mins followed by protein addition measured over 20 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50208428(CHEMBL3883981)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant GGT1 (unknown origin) using GGPP as substrate preincubated for 5 mins followed by protein addition measured over 20 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
King Fahd University Of Petroleum And Minerals

Curated by ChEMBL
LigandPNGBDBM50208432(CHEMBL3884346)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant GGT1 (unknown origin) using GGPP as substrate preincubated for 5 mins followed by protein addition measured over 20 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed