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Found 10 of ec50 for UniProtKB: P04694
TargetTyrosine aminotransferase(Rattus norvegicus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50272520((8S,9R,10S,11S,13S,14S,16S,17R)-9-fluoro-11-hydrox...)
Affinity DataEC50:  2nMAssay Description:Transactivation activity of tyrosine amino transferase in rat H4 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine aminotransferase(Rattus norvegicus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50272434((11beta,16beta)-9-Fluoro-11,21-dihydroxy-16-methyl...)
Affinity DataEC50:  5.30nMAssay Description:Transactivation activity of tyrosine amino transferase in rat H4 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine aminotransferase(Rattus norvegicus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50272521(Adamantan-1-yl-carbamic acid (8S,9R,10S,11S,13S,14...)
Affinity DataEC50:  9.80nMAssay Description:Transactivation activity of tyrosine amino transferase in rat H4 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine aminotransferase(Rattus norvegicus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50272523((11beta,16beta)-9-Fluoro-11,21-dihydroxy-16-methyl...)
Affinity DataEC50:  37.3nMAssay Description:Transactivation activity of tyrosine amino transferase in rat H4 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine aminotransferase(Rattus norvegicus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50272522((11beta,16beta)-9-Fluoro-11,21-dihydroxy-16-methyl...)
Affinity DataEC50:  70.3nMAssay Description:Transactivation activity of tyrosine amino transferase in rat H4 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine aminotransferase(Rattus norvegicus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50272400((8S,9R,10S,11S,13S,14S,16S,17R)-9-fluoro-11-hydrox...)
Affinity DataEC50:  117nMAssay Description:Transactivation activity of tyrosine amino transferase in rat H4 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine aminotransferase(Rattus norvegicus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50272493((8S,9R,10S,11S,13S,14S,16S,17R)-9-fluoro-11-hydrox...)
Affinity DataEC50:  156nMAssay Description:Transactivation activity of tyrosine amino transferase in rat H4 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine aminotransferase(Rattus norvegicus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50272435((11beta,16beta)-9-Fluoro-11,21-dihydroxy-16-methyl...)
Affinity DataEC50:  211nMAssay Description:Transactivation activity of tyrosine amino transferase in rat H4 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine aminotransferase(Rattus norvegicus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50272492((8S,9R,10S,11S,13S,14S,16S,17R)-9-fluoro-11-hydrox...)
Affinity DataEC50:  646nMAssay Description:Transactivation activity of tyrosine amino transferase in rat H4 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine aminotransferase(Rattus norvegicus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50272469((8S,9R,10S,11S,13S,14S,16S,17R)-9-fluoro-11-hydrox...)
Affinity DataEC50:  705nMAssay Description:Transactivation activity of tyrosine amino transferase in rat H4 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed