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Found 16 of ic50 for UniProtKB: A0A198XCR2
TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandPNGBDBM50212637(CHEMBL72046)
Affinity DataIC50:  2.85nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandPNGBDBM50212640(CHEMBL423309)
Affinity DataIC50:  2.89nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandPNGBDBM50212639(CHEMBL302241)
Affinity DataIC50:  2.90nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandPNGBDBM50212634(CHEMBL309009)
Affinity DataIC50:  5.23nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandPNGBDBM50212638(CHEMBL302512)
Affinity DataIC50:  8.64nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandPNGBDBM50212641(Brobactam)
Affinity DataIC50:  10.7nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandPNGBDBM50212646(CHEMBL72972)
Affinity DataIC50:  13.1nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandPNGBDBM50212642(CHEMBL70269)
Affinity DataIC50:  23.3nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandPNGBDBM50021959(CHEMBL777 | MM 14151 | US9120808, Clavulanic acid ...)
Affinity DataIC50:  30.1nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50:  33.3nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandPNGBDBM50212635(CHEMBL415266)
Affinity DataIC50:  50.7nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandPNGBDBM50212643(CHEMBL308516)
Affinity DataIC50:  56.1nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandPNGBDBM50212644(CHEMBL73450)
Affinity DataIC50:  63.7nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandPNGBDBM50212645(CHEMBL305908)
Affinity DataIC50:  65.9nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandPNGBDBM50212636(CHEMBL310221)
Affinity DataIC50:  80.5nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandPNGBDBM50021954((2S,5R)-3,3-Dimethyl-4,4,7-trioxo-4lambda*6*-thia-...)
Affinity DataIC50:  107nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails