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Found 4 of ic50 for UniProtKB: A0A0A7KLD0
TargetGlucocorticoid receptor(Canis lupus familiaris)
Oric Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM18627((10S,11S,14S,15S,17R)-17-[4-(dimethylamino)phenyl]...)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at GR in dog PBMC assessed as reduction in dexamethasone-induced FKBP5 gene expression incubated for 6 hrs by RT-qPCR methodMore data for this Ligand-Target Pair
TargetGlucocorticoid receptor(Canis lupus familiaris)
Oric Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50368933(CHEMBL4161754)
Affinity DataIC50:  25nMAssay Description:Antagonist activity at GR in dog PBMC assessed as reduction in dexamethasone-induced FKBP5 gene expression incubated for 6 hrs by RT-qPCR methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Canis lupus familiaris)
Oric Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM18627((10S,11S,14S,15S,17R)-17-[4-(dimethylamino)phenyl]...)
Affinity DataIC50:  33nMAssay Description:Antagonist activity at GR in dog PBMC assessed as reduction in dexamethasone-induced GILZ gene expression incubated for 6 hrs by RT-qPCR methodMore data for this Ligand-Target Pair
TargetGlucocorticoid receptor(Canis lupus familiaris)
Oric Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50368933(CHEMBL4161754)
Affinity DataIC50:  34nMAssay Description:Antagonist activity at GR in dog PBMC assessed as reduction in dexamethasone-induced GILZ gene expression incubated for 6 hrs by RT-qPCR methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed