Compile Data Set for Download or QSAR
maximum 50k data
Found 33 of ic50 for UniProtKB: A0A0S2Z448
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459727(CHEMBL4206834)
Affinity DataIC50:  57nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459737(CHEMBL4211204)
Affinity DataIC50:  82nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459731(CHEMBL4216416)
Affinity DataIC50:  120nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459738(CHEMBL4209820)
Affinity DataIC50:  140nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459730(CHEMBL4211714)
Affinity DataIC50:  149nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459747(CHEMBL4216933)
Affinity DataIC50:  341nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459735(CHEMBL4216170)
Affinity DataIC50:  369nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459726(CHEMBL4211962)
Affinity DataIC50:  372nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50576674(CHEMBL4850575)
Affinity DataIC50:  410nMAssay Description:Inhibition of AF9 YEATS domain (1 to 138 residues) (unknown origin) assessed as inhibition of probe-1 induced AF9 YEATS domain labelling incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50566890(CHEMBL4865432)
Affinity DataIC50:  729nMAssay Description:Inhibition of human His-AF9 YEATS domain and biotinylated H3K9ac peptide interaction by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459733(CHEMBL4209508)
Affinity DataIC50:  850nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50566877(CHEMBL4863719)
Affinity DataIC50:  984nMAssay Description:Inhibition of human His-AF9 YEATS domain and biotinylated H3K9ac peptide interaction by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459722(CHEMBL4204545)
Affinity DataIC50:  1.02E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459739(CHEMBL4204942)
Affinity DataIC50:  1.04E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459745(CHEMBL4210431)
Affinity DataIC50:  1.10E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459742(CHEMBL4204647)
Affinity DataIC50:  1.14E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459743(CHEMBL4209087)
Affinity DataIC50:  1.20E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459748(CHEMBL4213382)
Affinity DataIC50:  1.49E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459746(CHEMBL4212941)
Affinity DataIC50:  1.66E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50576675(CHEMBL4848627)
Affinity DataIC50:  1.74E+3nMAssay Description:Inhibition of AF9 YEATS domain (1 to 138 residues) (unknown origin) assessed as inhibition of probe-1 induced AF9 YEATS domain labelling incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459736(CHEMBL4216206)
Affinity DataIC50:  1.78E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50566867(CHEMBL4855926)
Affinity DataIC50:  1.85E+3nMAssay Description:Inhibition of human His-AF9 YEATS domain and biotinylated H3K9ac peptide interaction by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459729(CHEMBL4217882)
Affinity DataIC50:  2.37E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459732(CHEMBL4206070)
Affinity DataIC50:  3.49E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459734(CHEMBL4208554)
Affinity DataIC50:  4.11E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459740(CHEMBL4214833)
Affinity DataIC50:  4.29E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459724(CHEMBL4217790)
Affinity DataIC50:  4.66E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50566873(CHEMBL4859531)
Affinity DataIC50:  4.93E+3nMAssay Description:Inhibition of human His-AF9 YEATS domain and biotinylated H3K9ac peptide interaction by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459728(CHEMBL4205558)
Affinity DataIC50:  6.40E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459741(CHEMBL4209918)
Affinity DataIC50:  7.23E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459721(CHEMBL4213487)
Affinity DataIC50:  1.42E+4nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459725(CHEMBL4204221)
Affinity DataIC50:  2.43E+4nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459723(CHEMBL4218308)
Affinity DataIC50:  3.05E+4nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed