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Found 19 of ic50 for UniProtKB: P06869
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
University Of Michigan

LigandPNGBDBM92479(Tannic Acid, A | Tannic acid)
Affinity DataIC50:  4.10nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
University Of Michigan

LigandPNGBDBM50228412(CHEMBL393979 | methyl 1-(bis(4-acetamidophenoxy)ph...)
Affinity DataIC50:  8nMAssay Description:Inhibition of mouse uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
University Of Michigan

LigandPNGBDBM92485(CDE-066 | US9120744, CDE-066)
Affinity DataIC50:  10nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
University Of Michigan

LigandPNGBDBM50531924(CHEMBL4464577)
Affinity DataIC50:  10nMAssay Description:Inhibition of uPA in presence of 75% mouse serum measured immediatelyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
University Of Michigan

LigandPNGBDBM50531924(CHEMBL4464577)
Affinity DataIC50:  11nMAssay Description:Inhibition of uPA in presence of 75% mouse serum measured at 8 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
University Of Michigan

LigandPNGBDBM50531924(CHEMBL4464577)
Affinity DataIC50:  12nMAssay Description:Inhibition of uPA in presence of 75% mouse serum measured at 2 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
University Of Michigan

LigandPNGBDBM50228418(CHEMBL393591 | methyl 1-(diphenoxyphosphoryl)-2-(4...)
Affinity DataIC50:  32nMAssay Description:Inhibition of mouse uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
University Of Michigan

LigandPNGBDBM50531924(CHEMBL4464577)
Affinity DataIC50:  71nMAssay Description:Inhibition of uPA in presence of 75% mouse serum measured at 24 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
University Of Michigan

LigandPNGBDBM92486(CDE-082 | US9120744, CDE-082)
Affinity DataIC50:  79nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
University Of Michigan

LigandPNGBDBM92487(CDE-031 | US9120744, CDE-031)
Affinity DataIC50:  132nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
University Of Michigan

LigandPNGBDBM92482(CDE-008 | US9120744, CDE-008)
Affinity DataIC50:  162nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
University Of Michigan

LigandPNGBDBM50467212(CHEMBL4285028)
Affinity DataIC50:  410nMAssay Description:Inhibition of mouse uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
University Of Michigan

LigandPNGBDBM92483(CDE-034 | US9120744, CDE-034)
Affinity DataIC50:  644nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
University Of Michigan

LigandPNGBDBM92484(CDE-056 | US9120744, CDE-056)
Affinity DataIC50:  758nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
University Of Michigan

LigandPNGBDBM16173(3,5-diamino-6-chloro-N-(diaminomethylene)pyrazinam...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of mouse uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
University Of Michigan

LigandPNGBDBM50531924(CHEMBL4464577)
Affinity DataIC50:  3.28E+3nMAssay Description:Inhibition of the intrinsic peri-cellular uPA in mouse CT26 cells assessed as reduction in cell invasion measured every hour by transwell assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
University Of Michigan

LigandPNGBDBM50531926(CHEMBL4550668)
Affinity DataIC50:  5.02E+3nMAssay Description:Inhibition of the intrinsic peri-cellular uPA in mouse CT26 cells assessed as reduction in cell invasion measured every hour by transwell assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
University Of Michigan

LigandPNGBDBM50529246(CHEMBL4473654)
Affinity DataIC50:  1.42E+4nMAssay Description:Inhibition of mouse uPAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
University Of Michigan

LigandPNGBDBM50531925(CHEMBL4522772)
Affinity DataIC50:  3.94E+4nMAssay Description:Inhibition of the intrinsic peri-cellular uPA in mouse CT26 cells assessed as reduction in cell invasion measured every hour by transwell assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed