Compile Data Set for Download or QSAR
maximum 50k data
Found 14 of kd for UniProtKB: P30556
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50236697(5-L-isoleucineangiotensin II | 5-isoleucine-angiot...)
Affinity DataKd:  2nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50159215(CHEMBL3787375)
Affinity DataKd:  0.930nMAssay Description:Binding affinity to human AT1 receptor transfected in CHO cells co-expressing Galpha16-mtAEQ after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50052104(CHEMBL410812 | Sar-Arg-Val-Tyr-Asp-His-Apt-Phe)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50052103(CHEMBL217873 | Sar-Arg-Val-Tyr-Glu-His-Apt-Phe)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50052105(CHEMBL405938 | Sar-Arg-Val-Tyr-Cys-His-Pen-Phe)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50052106(CHEMBL406170 | Sar-Arg-Val-Tyr-Cys-His-Mpc-Phe)
Affinity DataKd:  2.30E+3nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50580361(CHEMBL5075338)
Affinity DataKd:  0.490nMAssay Description:Binding affinity to AT1R (unknown origin) expressed in Escherichia coli strain BL 21 (DE3) incubated for 20 mins by SDS PAGE analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50052101(2-({1-[2-{2-[2-{2-[5-Guanidino-2-(2-methylamino-ac...)
Affinity DataKd:  0.540nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50052109(CHEMBL412864 | Sar-Arg-Val-Tyr-Cys-His-Mpt-Phe)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50052102(CHEMBL414918 | Sar-Arg-Val-D-Tyr-Pro-His-Pro-Phe)
Affinity DataKd:  58nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50052110(CHEMBL216678 | Sar-Arg-Val-Tyr-Hcy-His-Mpt-Phe)
Affinity DataKd:  750nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50518054(CHEMBL4517561)
Affinity DataKd:  300nMAssay Description:Binding affinity to human AT1 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50048128(Asp-Arg-Val-Tyr-Val-His-Pro-Phe (Angiotensin II) |...)
Affinity DataKd:  1.60nMAssay Description:Binding affinity to human AT1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50052108(CHEMBL415025 | Sar-Arg-Val-Tyr-Hcy-His-Mpc-Phe)
Affinity DataKd:  20nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed