Compile Data Set for Download or QSAR
maximum 50k data
Found 54 of ec50 for UniProtKB: A0A024R328
LigandPNGBDBM50519087(CHEMBL3741746)
Affinity DataEC50:  0.190nMAssay Description:Agonist activity at Protein kinase C in human U1 cells infected with HIV-1 NL4-3 assessed as induction of HIV-1 p24 production after 72 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50519063(CHEMBL4587471)
Affinity DataEC50:  0.550nMAssay Description:Agonist activity at Protein kinase C in human U1 cells infected with HIV-1 NL4-3 assessed as induction of HIV-1 p24 production after 72 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50519068(CHEMBL4575056)
Affinity DataEC50:  0.600nMAssay Description:Agonist activity at Protein kinase C in human U1 cells infected with HIV-1 NL4-3 assessed as induction of HIV-1 p24 production after 72 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50495192(CHEMBL3105098)
Affinity DataEC50:  2.5nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50493441(CHEMBL2430122)
Affinity DataEC50:  2.90nMAssay Description:Activation of PKCdelta (unknown origin) using phosphatidylserine as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50495189(CHEMBL3105094)
Affinity DataEC50:  3.30nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50495197(CHEMBL3105027)
Affinity DataEC50:  3.70nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50495200(CHEMBL3105089)
Affinity DataEC50:  3.80nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50519085(CHEMBL4444766)
Affinity DataEC50: >3.90nMAssay Description:Agonist activity at Protein kinase C in human U1 cells infected with HIV-1 NL4-3 assessed as induction of HIV-1 p24 production after 72 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50470108(AGN 204332 | Ingenol Mebutate | PEP-005 | PEP005 |...)
Affinity DataEC50:  4.10nMAssay Description:Activation of PKCdelta (unknown origin) using phosphatidylserine as substrateMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50470108(AGN 204332 | Ingenol Mebutate | PEP-005 | PEP005 |...)
Affinity DataEC50:  4.10nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50495201(CHEMBL3105096)
Affinity DataEC50:  4.20nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50493442(CHEMBL2430115)
Affinity DataEC50:  4.5nMAssay Description:Activation of PKCdelta (unknown origin) using phosphatidylserine as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50493440(CHEMBL2430127)
Affinity DataEC50:  4.70nMAssay Description:Activation of PKCdelta (unknown origin) using phosphatidylserine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50493446(CHEMBL2430142)
Affinity DataEC50:  5.20nMAssay Description:Activation of PKCdelta (unknown origin) using phosphatidylserine as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50493443(CHEMBL2430141)
Affinity DataEC50:  5.30nMAssay Description:Activation of PKCdelta (unknown origin) using phosphatidylserine as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50493444(CHEMBL2430126)
Affinity DataEC50:  5.30nMAssay Description:Activation of PKCdelta (unknown origin) using phosphatidylserine as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50495191(CHEMBL2430121)
Affinity DataEC50:  6.10nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM239069(US9409931, 8)
Affinity DataEC50:  7nMpH: 7.4Assay Description:On the day at experiment Human Protein Kinase C delta (PKCδ, Millipore cat#14-504) was diluted in 20 mM HEPES, 0.03% Triton X-100. Amount of enz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50495188(CHEMBL3105106)
Affinity DataEC50:  8nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50099066(CHEMBL279115 | phorbol 13-acetate 12-myristate)
Affinity DataEC50:  9.5nMAssay Description:Activation of PKC in human platelet assessed as induction of platelet aggregation measured within 15 mins by tribidimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50493445(CHEMBL2430124)
Affinity DataEC50:  11nMAssay Description:Activation of PKCdelta (unknown origin) using phosphatidylserine as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50495199(CHEMBL3105102)
Affinity DataEC50:  11nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50495202(CHEMBL3105110)
Affinity DataEC50:  13nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50495196(CHEMBL3105095)
Affinity DataEC50:  13nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50495194(CHEMBL3105104)
Affinity DataEC50:  20nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50495190(CHEMBL3105092)
Affinity DataEC50:  26nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50470108(AGN 204332 | Ingenol Mebutate | PEP-005 | PEP005 |...)
Affinity DataEC50:  73nMAssay Description:Activation of PKC in human platelet assessed as induction of platelet aggregation measured within 15 mins by tribidimetric methodMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM239070(US9409931, 6)
Affinity DataEC50:  80nMpH: 7.4Assay Description:On the day at experiment Human Protein Kinase C delta (PKCδ, Millipore cat#14-504) was diluted in 20 mM HEPES, 0.03% Triton X-100. Amount of enz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM239071(US9409931, 7)
Affinity DataEC50:  154nMpH: 7.4Assay Description:On the day at experiment Human Protein Kinase C delta (PKCδ, Millipore cat#14-504) was diluted in 20 mM HEPES, 0.03% Triton X-100. Amount of enz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50495193(CHEMBL3105103)
Affinity DataEC50:  156nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50099066(CHEMBL279115 | phorbol 13-acetate 12-myristate)
Affinity DataEC50:  290nMAssay Description:Activation of PKCdelta (unknown origin) expressed in HEK293 cells harboring GFP-tagged RasGRP3 assessed as phosphorylation at ser299 residues after 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50368315(PROSTRATIN)
Affinity DataEC50:  910nMAssay Description:Activation of PKC in human platelet assessed as induction of platelet aggregation measured within 15 mins by tribidimetric methodMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50495195(CHEMBL3105026)
Affinity DataEC50:  988nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM239072(US9409931, 5)
Affinity DataEC50:  1.11E+3nMpH: 7.4Assay Description:On the day at experiment Human Protein Kinase C delta (PKCδ, Millipore cat#14-504) was diluted in 20 mM HEPES, 0.03% Triton X-100. Amount of enz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM50470110(CHEMBL4071723)
Affinity DataEC50:  5.04E+3nMAssay Description:Activation of PKC in human platelet assessed as induction of platelet aggregation measured within 15 mins by tribidimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50099066(CHEMBL279115 | phorbol 13-acetate 12-myristate)
Affinity DataEC50:  5.17E+3nMAssay Description:Binding affinity to GST-tagged PKCdelta expressed in Escherichia coli BL21(DE3) by fluorescence quenchingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50470109(CHEMBL4104319)
Affinity DataEC50:  6.08E+3nMAssay Description:Activation of PKC in human platelet assessed as induction of platelet aggregation measured within 15 mins by tribidimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50307105(1,2-dioleoyl-sn-glycerol | CHEMBL590047)
Affinity DataEC50:  7.49E+3nMAssay Description:Binding affinity to GST-tagged PKCdelta expressed in Escherichia coli BL21(DE3) by fluorescence quenchingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50280749(CHEMBL4169454)
Affinity DataEC50:  8.03E+3nMAssay Description:Activation of PKCdelta (unknown origin) expressed in human LNCAP cells harboring GFP-tagged RasGRP1 assessed as phosphorylation at ser299 residues af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50280749(CHEMBL4169454)
Affinity DataEC50:  8.28E+3nMAssay Description:Activation of PKCdelta (unknown origin) expressed in human LNCAP cells harboring GFP-tagged RasGRP3 assessed as phosphorylation at ser299 residues af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50307103((1E,4Z,6E)-7-(4-(Hexadecyloxy)-3-methoxyphenyl)-5-...)
Affinity DataEC50:  8.69E+3nMAssay Description:Binding affinity to GST-tagged PKCdelta expressed in Escherichia coli BL21(DE3) by fluorescence quenchingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50307104((1E,4Z,6E)-5-Hydroxy-1,7-bis(3-methoxy-4-(octyloxy...)
Affinity DataEC50:  8.98E+3nMAssay Description:Binding affinity to GST-tagged PKCdelta expressed in Escherichia coli BL21(DE3) by fluorescence quenchingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50495198(CHEMBL3105088)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50067040(((E,E)-1,7-bis(4-hydroxy-3-methoxyphenyl)-1,6-hept...)
Affinity DataEC50:  1.07E+4nMAssay Description:Binding affinity to GST-tagged PKCdelta expressed in Escherichia coli BL21(DE3) by fluorescence quenchingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50163745(4,40-(1E,10E)-2,20-(Isoxazole-3,5-diyl)bis(ethene-...)
Affinity DataEC50:  1.16E+4nMAssay Description:Binding affinity to PKCdelta C1B subdomain after 1 hr by fluorescence quenching analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50067030((1E,4Z,6E)-1,7-Bis-(3,4-dihydroxy-phenyl)-5-hydrox...)
Affinity DataEC50:  1.25E+4nMAssay Description:Binding affinity to GST-tagged PKCdelta expressed in Escherichia coli BL21(DE3) by fluorescence quenchingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50280749(CHEMBL4169454)
Affinity DataEC50:  1.26E+4nMAssay Description:Activation of PKCdelta (unknown origin) expressed in HEK293 cells harboring GFP-tagged RasGRP1 assessed as phosphorylation at ser299 residues after 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50163748((E)-3,5-Bis[beta-(4-Hydroxy-3-methoxyphenyl)-ethen...)
Affinity DataEC50:  1.50E+4nMAssay Description:Binding affinity to PKCdelta C1B subdomain after 1 hr by fluorescence quenching analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50015677((S)-1-hydroxymethyl-2-octanoyloxy-ethyl ester | 1,...)
Affinity DataEC50:  1.62E+4nMAssay Description:Binding affinity to GST-tagged PKCdelta expressed in Escherichia coli BL21(DE3) by fluorescence quenchingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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