Compile Data Set for Download or QSAR
maximum 50k data
Found 48 Enz. Inhib. hit(s) with all data for entry = 50019273
TargetD(4) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203383(CHEMBL228972 | N-(1-benzylpiperidin-4-yl)-2-naphth...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203374(CHEMBL234825 | naphthalene-2-carboxylic acid [1-(3...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203397(CHEMBL234645 | N-(1-(3-methoxybenzyl)piperidin-4-y...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203376(CHEMBL234826 | naphthalene-2-carboxylic acid [1-(4...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203377(CHEMBL234647 | naphthalene-2-carboxylic acid [1-(2...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203392(CHEMBL234646 | N-(1-(4-methoxybenzyl)piperidin-4-y...)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203373(CHEMBL234472 | N-(1-(4-bromobenzyl)piperidin-4-yl)...)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203382(CHEMBL395867 | N-(1-(3-bromobenzyl)piperidin-4-yl)...)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203378(CHEMBL233581 | N-(1-(4-chlorobenzyl)piperidin-4-yl...)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203388(CHEMBL234641 | N-(1-(4-chlorobenzyl)piperidin-4-yl...)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50203383(CHEMBL228972 | N-(1-benzylpiperidin-4-yl)-2-naphth...)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203394(CHEMBL234643 | N-(1-(4-bromobenzyl)piperidin-4-yl)...)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50203382(CHEMBL395867 | N-(1-(3-bromobenzyl)piperidin-4-yl)...)
Affinity DataKi:  53nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203389(CHEMBL233580 | N-(1-(3-chlorobenzyl)piperidin-4-yl...)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203393(CHEMBL395631 | N-(1-(3-bromobenzyl)piperidin-4-yl)...)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203391(CHEMBL233578 | naphthalene-1-carboxylic acid [1-(4...)
Affinity DataKi:  69nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203384(CHEMBL233404 | naphthalene-1-carboxylic acid [1-(3...)
Affinity DataKi:  77nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203386(CHEMBL430167 | N-(1-(4-(trifluoromethyl)benzyl)pip...)
Affinity DataKi:  84nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50203374(CHEMBL234825 | naphthalene-2-carboxylic acid [1-(3...)
Affinity DataKi:  87nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203385(CHEMBL234824 | N-(1-(4-(trifluoromethyl)benzyl)pip...)
Affinity DataKi:  96nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203381(CHEMBL234473 | N-(1-(3-(trifluoromethyl)benzyl)pip...)
Affinity DataKi:  103nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203398(CHEMBL234640 | N-(1-(3-chlorobenzyl)piperidin-4-yl...)
Affinity DataKi:  116nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203371(CHEMBL398990 | N-(1-(3-(trifluoromethyl)benzyl)pip...)
Affinity DataKi:  119nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50203389(CHEMBL233580 | N-(1-(3-chlorobenzyl)piperidin-4-yl...)
Affinity DataKi:  133nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50203399(CHEMBL233579 | N-(1-(2-chlorobenzyl)piperidin-4-yl...)
Affinity DataKi:  133nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50203392(CHEMBL234646 | N-(1-(4-methoxybenzyl)piperidin-4-y...)
Affinity DataKi:  151nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203372(CHEMBL395632 | naphthalene-1-carboxylic acid [1-(2...)
Affinity DataKi:  155nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50203397(CHEMBL234645 | N-(1-(3-methoxybenzyl)piperidin-4-y...)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203375(CHEMBL229019 | N-(1-benzylpiperidin-4-yl)-1-naphth...)
Affinity DataKi:  162nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203379(CHEMBL434583 | N-(1-(3-methoxybenzyl)piperidin-4-y...)
Affinity DataKi:  168nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50203377(CHEMBL234647 | naphthalene-2-carboxylic acid [1-(2...)
Affinity DataKi:  175nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203395(CHEMBL234644 | N-(1-(4-nitrobenzyl)piperidin-4-yl)...)
Affinity DataKi:  181nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50203376(CHEMBL234826 | naphthalene-2-carboxylic acid [1-(4...)
Affinity DataKi:  222nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203396(CHEMBL233403 | N-(1-(4-methoxybenzyl)piperidin-4-y...)
Affinity DataKi:  223nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50203373(CHEMBL234472 | N-(1-(4-bromobenzyl)piperidin-4-yl)...)
Affinity DataKi:  223nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50203380(CHEMBL232197 | N-(1-(perfluorobenzyl)piperidin-4-y...)
Affinity DataKi:  228nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50203378(CHEMBL233581 | N-(1-(4-chlorobenzyl)piperidin-4-yl...)
Affinity DataKi:  242nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50203395(CHEMBL234644 | N-(1-(4-nitrobenzyl)piperidin-4-yl)...)
Affinity DataKi:  278nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203370(CHEMBL234827 | N-(1-(pyridin-2-ylmethyl)piperidin-...)
Affinity DataKi:  299nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203390(CHEMBL394042 | N-(1-(pyridin-3-ylmethyl)piperidin-...)
Affinity DataKi:  326nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203400(CHEMBL233214 | N-(1-(2-chlorobenzyl)piperidin-4-yl...)
Affinity DataKi:  329nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50203393(CHEMBL395631 | N-(1-(3-bromobenzyl)piperidin-4-yl)...)
Affinity DataKi:  462nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50203390(CHEMBL394042 | N-(1-(pyridin-3-ylmethyl)piperidin-...)
Affinity DataKi:  524nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50203370(CHEMBL234827 | N-(1-(pyridin-2-ylmethyl)piperidin-...)
Affinity DataKi:  545nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50203387(CHEMBL234001 | N-(1-(pyridin-4-ylmethyl)piperidin-...)
Affinity DataKi:  695nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50203375(CHEMBL229019 | N-(1-benzylpiperidin-4-yl)-1-naphth...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203383(CHEMBL228972 | N-(1-benzylpiperidin-4-yl)-2-naphth...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2L receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50203375(CHEMBL229019 | N-(1-benzylpiperidin-4-yl)-1-naphth...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2L receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed