Compile Data Set for Download or QSAR
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Found 9 Enz. Inhib. hit(s) with all data for entry = 50034147
TargetCytohesin-3(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50357881(CHEMBL1916340)
Affinity DataKd:  140nMAssay Description:Binding affinity to recombinant rat brain Grp1 PH domain (amino acids 1 to 120) after 10 mins by pull-down assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target1-phosphatidylinositol 4,5-bisphosphate phosphodiesterase delta-1(Homo sapiens (Human))
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50357881(CHEMBL1916340)
Affinity DataKd:  250nMAssay Description:Binding affinity to PLCdelta1 PH domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytohesin-3(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50357881(CHEMBL1916340)
Affinity DataKd:  300nMAssay Description:Binding affinity to recombinant rat brain Grp1 PH domain (amino acids 1 to 120) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target1-phosphatidylinositol 4,5-bisphosphate phosphodiesterase delta-1(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50357881(CHEMBL1916340)
Affinity DataKd: >5.00E+3nMAssay Description:Binding affinity to recombinant rat brain PLCdelta1 PH domain (amino acids 11 to 140) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytohesin-3(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50075651(1D-myo-inositol 1,3,4,5-tetrakis(dihydrogen phosph...)
Affinity DataKd:  100nMAssay Description:Binding affinity to recombinant rat brain Grp1 PH domain (amino acids 1 to 120) after 10 mins by pull-down assayMore data for this Ligand-Target Pair
Target1-phosphatidylinositol 4,5-bisphosphate phosphodiesterase delta-1(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50357882(CHEMBL1916341)
Affinity DataKd:  2.20E+3nMAssay Description:Binding affinity to recombinant rat brain PLCdelta1 PH domain (amino acids 11 to 140) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytohesin-3(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50357883(CHEMBL1916342)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to recombinant rat brain Grp1 PH domain (amino acids 1 to 120) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target1-phosphatidylinositol 4,5-bisphosphate phosphodiesterase delta-1(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50357883(CHEMBL1916342)
Affinity DataKd: >5.00E+3nMAssay Description:Binding affinity to recombinant rat brain PLCdelta1 PH domain (amino acids 11 to 140) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytohesin-3(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50357882(CHEMBL1916341)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to recombinant rat brain Grp1 PH domain (amino acids 1 to 120) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed