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Found 25 Enz. Inhib. hit(s) with all data for entry = 50008568
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£T Bonn

Curated by ChEMBL
LigandPNGBDBM50520503(CHEMBL4471610)
Affinity DataKi:  609nMAssay Description:Displacement of [3H]PSB-11 from human A3 adenosine receptor expressed in CHO cell membranes incubated for 60 mins by liquid scintillation counting me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£T Bonn

Curated by ChEMBL
LigandPNGBDBM50483929(Archazolid F | CHEBI:67525)
Affinity DataKi:  859nMAssay Description:Displacement of [3H]PSB-11 from human A3 adenosine receptor expressed in CHO cell membranes incubated for 60 mins by liquid scintillation counting me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£T Bonn

Curated by ChEMBL
LigandPNGBDBM50178305(ARCHAZOLID A)
Affinity DataKi:  967nMAssay Description:Displacement of [3H]PSB-11 from human A3 adenosine receptor expressed in CHO cell membranes incubated for 60 mins by liquid scintillation counting me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£T Bonn

Curated by ChEMBL
LigandPNGBDBM50064186((3Z,5E,7R,8S,9S,11E,13E,15S,16R)-16-{(2S,3R,4S)-4-...)
Affinity DataKi:  1.08E+3nMAssay Description:Displacement of [3H]PSB-11 from human A3 adenosine receptor expressed in CHO cell membranes incubated for 60 mins by liquid scintillation counting me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£T Bonn

Curated by ChEMBL
LigandPNGBDBM50520505(CHEMBL4593430)
Affinity DataKi:  1.14E+3nMAssay Description:Displacement of [3H]PSB-11 from human A3 adenosine receptor expressed in CHO cell membranes incubated for 60 mins by liquid scintillation counting me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£T Bonn

Curated by ChEMBL
LigandPNGBDBM50483928(ARCHAZOLID B)
Affinity DataKi:  1.18E+3nMAssay Description:Displacement of [3H]PSB-11 from human A3 adenosine receptor expressed in CHO cell membranes incubated for 60 mins by liquid scintillation counting me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£T Bonn

Curated by ChEMBL
LigandPNGBDBM50520502(CHEMBL4447903)
Affinity DataKi:  1.38E+3nMAssay Description:Displacement of [3H]PSB-11 from human A3 adenosine receptor expressed in CHO cell membranes incubated for 60 mins by liquid scintillation counting me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£T Bonn

Curated by ChEMBL
LigandPNGBDBM50520501(CHEMBL4549217)
Affinity DataKi:  1.61E+3nMAssay Description:Displacement of [3H]PSB-11 from human A3 adenosine receptor expressed in CHO cell membranes incubated for 60 mins by liquid scintillation counting me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Universit£T Bonn

Curated by ChEMBL
LigandPNGBDBM50178305(ARCHAZOLID A)
Affinity DataIC50:  86nMAssay Description:Inhibition of human P2X3 assessed as reduction in agonist-induced intracellular Ca2+ concentration pre-incubated for 30 mins before agonist addition ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Universit£T Bonn

Curated by ChEMBL
LigandPNGBDBM50483928(ARCHAZOLID B)
Affinity DataIC50:  316nMAssay Description:Inhibition of human leukocyte elastase assessed as reduction in pNA release using chromogenic MeO-Suc-Ala-Ala-Pro-Val-pNA substrate measured over 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Universit£T Bonn

Curated by ChEMBL
LigandPNGBDBM50178305(ARCHAZOLID A)
Affinity DataIC50:  352nMAssay Description:Inhibition of human leukocyte elastase assessed as reduction in pNA release using chromogenic MeO-Suc-Ala-Ala-Pro-Val-pNA substrate measured over 10 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Universit£T Bonn

Curated by ChEMBL
LigandPNGBDBM50483928(ARCHAZOLID B)
Affinity DataIC50:  353nMAssay Description:Inhibition of human P2X3 assessed as reduction in agonist-induced intracellular Ca2+ concentration pre-incubated for 30 mins before agonist addition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Universit£T Bonn

Curated by ChEMBL
LigandPNGBDBM50483929(Archazolid F | CHEBI:67525)
Affinity DataIC50:  438nMAssay Description:Inhibition of human P2X3 assessed as reduction in agonist-induced intracellular Ca2+ concentration pre-incubated for 30 mins before agonist addition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Universit£T Bonn

Curated by ChEMBL
LigandPNGBDBM50520504(CHEMBL4460252)
Affinity DataIC50:  595nMAssay Description:Inhibition of human leukocyte elastase assessed as reduction in pNA release using chromogenic MeO-Suc-Ala-Ala-Pro-Val-pNA substrate measured over 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Universit£T Bonn

Curated by ChEMBL
LigandPNGBDBM50520505(CHEMBL4593430)
Affinity DataIC50:  648nMAssay Description:Inhibition of human P2X3 assessed as reduction in agonist-induced intracellular Ca2+ concentration pre-incubated for 30 mins before agonist addition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Universit£T Bonn

Curated by ChEMBL
LigandPNGBDBM50520505(CHEMBL4593430)
Affinity DataIC50:  721nMAssay Description:Inhibition of human leukocyte elastase assessed as reduction in pNA release using chromogenic MeO-Suc-Ala-Ala-Pro-Val-pNA substrate measured over 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Universit£T Bonn

Curated by ChEMBL
LigandPNGBDBM50064186((3Z,5E,7R,8S,9S,11E,13E,15S,16R)-16-{(2S,3R,4S)-4-...)
Affinity DataIC50:  755nMAssay Description:Inhibition of human P2X3 assessed as reduction in agonist-induced intracellular Ca2+ concentration pre-incubated for 30 mins before agonist addition ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Universit£T Bonn

Curated by ChEMBL
LigandPNGBDBM50483929(Archazolid F | CHEBI:67525)
Affinity DataIC50:  830nMAssay Description:Inhibition of human leukocyte elastase assessed as reduction in pNA release using chromogenic MeO-Suc-Ala-Ala-Pro-Val-pNA substrate measured over 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Universit£T Bonn

Curated by ChEMBL
LigandPNGBDBM50520503(CHEMBL4471610)
Affinity DataIC50:  1.31E+3nMAssay Description:Inhibition of human P2X3 assessed as reduction in agonist-induced intracellular Ca2+ concentration pre-incubated for 30 mins before agonist addition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Universit£T Bonn

Curated by ChEMBL
LigandPNGBDBM50520502(CHEMBL4447903)
Affinity DataIC50:  1.54E+3nMAssay Description:Inhibition of human leukocyte elastase assessed as reduction in pNA release using chromogenic MeO-Suc-Ala-Ala-Pro-Val-pNA substrate measured over 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Universit£T Bonn

Curated by ChEMBL
LigandPNGBDBM50520504(CHEMBL4460252)
Affinity DataIC50: >2.00E+3nMAssay Description:Inhibition of human P2X3 assessed as reduction in agonist-induced intracellular Ca2+ concentration pre-incubated for 30 mins before agonist addition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Universit£T Bonn

Curated by ChEMBL
LigandPNGBDBM50520501(CHEMBL4549217)
Affinity DataIC50:  2.34E+3nMAssay Description:Inhibition of human leukocyte elastase assessed as reduction in pNA release using chromogenic MeO-Suc-Ala-Ala-Pro-Val-pNA substrate measured over 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Universit£T Bonn

Curated by ChEMBL
LigandPNGBDBM50520503(CHEMBL4471610)
Affinity DataIC50:  5.85E+3nMAssay Description:Inhibition of human leukocyte elastase assessed as reduction in pNA release using chromogenic MeO-Suc-Ala-Ala-Pro-Val-pNA substrate measured over 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Universit£T Bonn

Curated by ChEMBL
LigandPNGBDBM50520501(CHEMBL4549217)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human P2X3 assessed as reduction in agonist-induced intracellular Ca2+ concentration pre-incubated for 30 mins before agonist addition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Universit£T Bonn

Curated by ChEMBL
LigandPNGBDBM50520502(CHEMBL4447903)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human P2X3 assessed as reduction in agonist-induced intracellular Ca2+ concentration pre-incubated for 30 mins before agonist addition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed