Compile Data Set for Download or QSAR
maximum 50k data
Found 245 of ec50 data for polymerid = 2268
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22376((3aS,6aR)-4-cyclohexyl-5-[(4E)-oct-4-en-4-yl]-N-ph...)
Affinity DataEC50:  10nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22391((3aS,6aR)-N-(2,3-dimethylphenyl)-5-hexyl-4-phenyl-...)
Affinity DataEC50:  11nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22381((3aS,6aR)-5-[(6E)-dodec-6-en-6-yl]-N,4-diphenyl-1,...)
Affinity DataEC50:  14nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22375((3aS,6aR)-4-butyl-5-[(4E)-oct-4-en-4-yl]-N-phenyl-...)
Affinity DataEC50:  30nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM50418303(CHEMBL1765959)
Affinity DataEC50:  31.6nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM50418304(CHEMBL1765953)
Affinity DataEC50:  39.8nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22385((3aS,6aR)-5-hexyl-N,4-diphenyl-1,2,3,3a,6,6a-hexah...)
Affinity DataEC50:  39.8nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22385((3aS,6aR)-5-hexyl-N,4-diphenyl-1,2,3,3a,6,6a-hexah...)
Affinity DataEC50:  43nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22373((3aS,6aR)-5-[(4E)-oct-4-en-4-yl]-N,4-diphenyl-1,2,...)
Affinity DataEC50:  54nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM50418308(CHEMBL1765933)
Affinity DataEC50:  63.1nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM50418307(CHEMBL1765934)
Affinity DataEC50:  63.1nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM50418306(CHEMBL1765955)
Affinity DataEC50:  63.1nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM50418305(CHEMBL1765960)
Affinity DataEC50:  63.1nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM50418309(CHEMBL1765956)
Affinity DataEC50:  63.1nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM50418310(CHEMBL1765962)
Affinity DataEC50:  79.4nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM50418311(CHEMBL1765931)
Affinity DataEC50:  79.4nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM28650(ethyl 2-[(2-{[(4-ethylphenyl)carbamoyl]methyl}-1-o...)
Affinity DataEC50:  110nMAssay Description:The assay was to monitor the SF-1 activation state via co-transfection of CHO-K1 cells with a plasmid encoding a Gal4-SF-1 chimerical transcription f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22388((3aS,6aR)-N,4,5-triphenyl-1,2,3,3a,6,6a-hexahydrop...)
Affinity DataEC50:  120nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM50418313(CHEMBL1765945)
Affinity DataEC50:  126nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM39548((2-phenyl-1,3-thiazol-4-yl)methyl 1-methylpyrrole-...)
Affinity DataEC50:  129nMAssay Description:Source (MLSCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute, TSRI Assay ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22379((3aS,6aR)-4-(naphthalen-2-yl)-5-[(4E)-oct-4-en-4-y...)
Affinity DataEC50:  130nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22383((3aS,6aR)-5-(decan-2-yl)-N,4-diphenyl-1,2,3,3a,6,6...)
Affinity DataEC50:  130nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22382((3aS,6aR)-5-(hexan-2-yl)-N,4-diphenyl-1,2,3,3a,6,6...)
Affinity DataEC50:  130nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM39480(2-(1-tert-butyl-4-keto-pyrazolo[3,4-d]pyrimidin-5-...)
Affinity DataEC50:  138nMAssay Description:Source (MLSCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute, TSRI Assay ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM39527(MLS000070707 | N-(6-ethoxy-1,3-benzothiazol-2-yl)-...)
Affinity DataEC50:  140nMAssay Description:Source (MLSCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute, TSRI Assay ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22378((3aS,6aR)-4-(3-methoxyphenyl)-5-[(4E)-oct-4-en-4-y...)
Affinity DataEC50:  140nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM50418314(CHEMBL1765954)
Affinity DataEC50:  158nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22373((3aS,6aR)-5-[(4E)-oct-4-en-4-yl]-N,4-diphenyl-1,2,...)
Affinity DataEC50:  158nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM50418300(CHEMBL1765941)
Affinity DataEC50:  158nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM50418315(CHEMBL1765936)
Affinity DataEC50:  158nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM39428(5-Methyl-furan-2-carboxylic acid (5-benzyl-thiazol...)
Affinity DataEC50:  168nMAssay Description:Source (MLSCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute, TSRI Assay ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22377((3aS,6aR)-4-(4-bromophenyl)-5-[(4E)-oct-4-en-4-yl]...)
Affinity DataEC50:  170nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22386((3aS,6aR)-5-cyclohexyl-N,4-diphenyl-1,2,3,3a,6,6a-...)
Affinity DataEC50:  180nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM39426(7-amino-3-phenyl-6-pyrazolo[1,5-a]pyrimidinecarbox...)
Affinity DataEC50:  183nMAssay Description:Source (MLSCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute, TSRI Assay ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM28649(ethyl 2-[(2-{[(4-ethoxyphenyl)carbamoyl]methyl}-1-...)
Affinity DataEC50:  190nMAssay Description:The assay was to monitor the SF-1 activation state via co-transfection of CHO-K1 cells with a plasmid encoding a Gal4-SF-1 chimerical transcription f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM39531(8-methyl-2-phenyl-imidazo[1,2-a]pyridine | 8-methy...)
Affinity DataEC50:  190nMAssay Description:Source (MLSCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute, TSRI Assay ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM28648(ethyl 2-{[1-oxo-2-({[4-(trifluoromethoxy)phenyl]ca...)
Affinity DataEC50:  200nMAssay Description:The assay was to monitor the SF-1 activation state via co-transfection of CHO-K1 cells with a plasmid encoding a Gal4-SF-1 chimerical transcription f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM50418320(CHEMBL1765927)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM50418319(CHEMBL1765930)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM50418318(CHEMBL1765942)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM50418316(CHEMBL1765966)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM28647(ethyl 2-[(2-{[(4-methoxyphenyl)carbamoyl]methyl}-1...)
Affinity DataEC50:  200nMAssay Description:The assay was to monitor the SF-1 activation state via co-transfection of CHO-K1 cells with a plasmid encoding a Gal4-SF-1 chimerical transcription f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM50418317(CHEMBL1765950)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM39543(3-(3-methoxyphenyl)-5-(2-thienyl)-1,2,4-oxadiazole...)
Affinity DataEC50:  226nMAssay Description:Source (MLSCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute, TSRI Assay ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM39565(2-(2-chlorophenyl)-5-(4-chlorophenyl)-1,3,4-oxadia...)
Affinity DataEC50:  233nMAssay Description:Source (MLSCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute, TSRI Assay ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM50418302(CHEMBL1765929)
Affinity DataEC50:  251nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM50418321(CHEMBL1765963)
Affinity DataEC50:  251nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM50418322(CHEMBL1765948)
Affinity DataEC50:  251nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM39534(1-azepanyl-[4-(5-phenyl-1,3,4-oxadiazol-2-yl)pheny...)
Affinity DataEC50:  252nMAssay Description:Source (MLSCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute, TSRI Assay ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM39537(MLS000077996 | N-[5-(1-adamantyl)-1,3,4-thiadiazol...)
Affinity DataEC50:  257nMAssay Description:Source (MLSCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute, TSRI Assay ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
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