Compile Data Set for Download or QSAR
maximum 50k data
Found 212 of ec50 data for polymerid = 3035
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50082078(CHEMBL3422411)
Affinity DataEC50:  0.00600nMAssay Description:Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50508242(CHEMBL4539775)
Affinity DataEC50:  0.0220nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50392485(CHEMBL2152055)
Affinity DataEC50:  0.0230nMAssay Description:Agonist activity at human OT7T175 assessed as increase in intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50508234(CHEMBL4533110)
Affinity DataEC50:  0.0240nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50508221(CHEMBL4462883)
Affinity DataEC50:  0.0280nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50392490(CHEMBL2152060)
Affinity DataEC50:  0.0290nMAssay Description:Agonist activity at human OT7T175 assessed as increase in intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50508225(CHEMBL4528114)
Affinity DataEC50:  0.0370nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50392486(CHEMBL2152056)
Affinity DataEC50:  0.0390nMAssay Description:Agonist activity at human OT7T175 assessed as increase in intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50392402(CHEMBL2151643)
Affinity DataEC50:  0.0410nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM26349((2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-amino-3-(4-hydroxyp...)
Affinity DataEC50:  0.0490nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50392405(CHEMBL2151646)
Affinity DataEC50:  0.0500nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50442964(CHEMBL3085809)
Affinity DataEC50:  0.0570nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50508241(CHEMBL4451244)
Affinity DataEC50:  0.0580nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50392401(CHEMBL2151642)
Affinity DataEC50:  0.0650nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50392488(CHEMBL2152058)
Affinity DataEC50:  0.0650nMAssay Description:Agonist activity at human OT7T175 assessed as increase in intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM26349((2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-amino-3-(4-hydroxyp...)
Affinity DataEC50:  0.0650nMAssay Description:Agonist activity at human OT7T175 assessed as increase in intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50508220(CHEMBL4541289)
Affinity DataEC50:  0.0680nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50082074(CHEMBL3422408)
Affinity DataEC50:  0.0700nMAssay Description:Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50082073(CHEMBL3422407)
Affinity DataEC50:  0.0700nMAssay Description:Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50392413(CHEMBL2151654)
Affinity DataEC50:  0.0720nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50196431(CHEMBL3949159)
Affinity DataEC50:  0.0730nMAssay Description:Agonist activity at human KISS1R expressed in CHO/dhfr cells assessed as increase in intracellular Ca2+ levels measured for 180 secs by Fluo 3-AM dye...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50082068(CHEMBL3422414)
Affinity DataEC50:  0.0800nMAssay Description:Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50045513(Kisspeptin-10)
Affinity DataEC50:  0.0870nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50392412(CHEMBL2151653)
Affinity DataEC50:  0.0980nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50082067(CHEMBL3422413)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50392409(CHEMBL2151650)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50392411(CHEMBL2151652)
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50508237(CHEMBL4473151)
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50508233(CHEMBL4584512)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50508236(CHEMBL4563528)
Affinity DataEC50:  0.130nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50508231(CHEMBL4459547)
Affinity DataEC50:  0.130nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50392491(CHEMBL2152061)
Affinity DataEC50:  0.130nMAssay Description:Agonist activity at human OT7T175 assessed as increase in intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50392408(CHEMBL2151649)
Affinity DataEC50:  0.130nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50392492(CHEMBL2152062)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity at human OT7T175 assessed as increase in intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50508218(CHEMBL4536531)
Affinity DataEC50:  0.160nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50508230(CHEMBL4439387)
Affinity DataEC50:  0.170nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50508224(CHEMBL4470916)
Affinity DataEC50:  0.230nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50392410(CHEMBL2151651)
Affinity DataEC50:  0.240nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50392407(CHEMBL2151648)
Affinity DataEC50:  0.240nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50508223(CHEMBL4538305)
Affinity DataEC50:  0.240nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50442961(CHEMBL3086284)
Affinity DataEC50:  0.270nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50392482(CHEMBL2152052)
Affinity DataEC50:  0.270nMAssay Description:Agonist activity at human OT7T175 assessed as increase in intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50508222(CHEMBL4468499)
Affinity DataEC50:  0.270nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50392484(CHEMBL2152054)
Affinity DataEC50:  0.290nMAssay Description:Agonist activity at human OT7T175 assessed as increase in intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50045506(CHEMBL3314223)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at human KISS1R transfected in CHO cells assessed as intracellular calcium flux after 24 hrs by functional FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50045500(CHEMBL3314217)
Affinity DataEC50:  0.310nMAssay Description:Agonist activity at human KISS1R transfected in CHO cells assessed as intracellular calcium flux after 24 hrs by functional FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50392487(CHEMBL2152057)
Affinity DataEC50:  0.320nMAssay Description:Agonist activity at human OT7T175 assessed as increase in intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50508228(CHEMBL4557192)
Affinity DataEC50:  0.330nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50045507(CHEMBL3314224)
Affinity DataEC50:  0.330nMAssay Description:Agonist activity at human KISS1R expressed in CHO/dhfr cells assessed as increase in intracellular Ca2+ levels measured for 180 secs by Fluo 3-AM dye...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50045507(CHEMBL3314224)
Affinity DataEC50:  0.330nMAssay Description:Agonist activity at human KISS1R transfected in CHO cells assessed as intracellular calcium flux after 24 hrs by functional FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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