Affinity DataEC50: 0.00600nMAssay Description:Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0220nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0230nMAssay Description:Agonist activity at human OT7T175 assessed as increase in intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0240nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0280nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0290nMAssay Description:Agonist activity at human OT7T175 assessed as increase in intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0370nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0390nMAssay Description:Agonist activity at human OT7T175 assessed as increase in intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0410nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0490nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0500nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0570nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0580nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0650nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0650nMAssay Description:Agonist activity at human OT7T175 assessed as increase in intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0650nMAssay Description:Agonist activity at human OT7T175 assessed as increase in intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0680nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0700nMAssay Description:Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0700nMAssay Description:Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0720nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0730nMAssay Description:Agonist activity at human KISS1R expressed in CHO/dhfr cells assessed as increase in intracellular Ca2+ levels measured for 180 secs by Fluo 3-AM dye...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0800nMAssay Description:Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0870nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0980nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 0.100nMAssay Description:Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.100nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 0.110nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 0.110nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Affinity DataEC50: 0.120nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Affinity DataEC50: 0.130nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Affinity DataEC50: 0.130nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Affinity DataEC50: 0.130nMAssay Description:Agonist activity at human OT7T175 assessed as increase in intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.130nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 0.150nMAssay Description:Agonist activity at human OT7T175 assessed as increase in intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.160nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Affinity DataEC50: 0.170nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Affinity DataEC50: 0.230nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Affinity DataEC50: 0.240nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 0.240nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 0.240nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Affinity DataEC50: 0.270nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Affinity DataEC50: 0.270nMAssay Description:Agonist activity at human OT7T175 assessed as increase in intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.270nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Affinity DataEC50: 0.290nMAssay Description:Agonist activity at human OT7T175 assessed as increase in intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.300nMAssay Description:Agonist activity at human KISS1R transfected in CHO cells assessed as intracellular calcium flux after 24 hrs by functional FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.310nMAssay Description:Agonist activity at human KISS1R transfected in CHO cells assessed as intracellular calcium flux after 24 hrs by functional FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.320nMAssay Description:Agonist activity at human OT7T175 assessed as increase in intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.330nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
Affinity DataEC50: 0.330nMAssay Description:Agonist activity at human KISS1R expressed in CHO/dhfr cells assessed as increase in intracellular Ca2+ levels measured for 180 secs by Fluo 3-AM dye...More data for this Ligand-Target Pair
Affinity DataEC50: 0.330nMAssay Description:Agonist activity at human KISS1R transfected in CHO cells assessed as intracellular calcium flux after 24 hrs by functional FLIPR assayMore data for this Ligand-Target Pair