TargetB2 bradykinin receptor(Homo sapiens (Human))
National Institute Of Neuroscienc
Curated by ChEMBL
National Institute Of Neuroscienc
Curated by ChEMBL
Affinity DataEC50: 0.0339nMAssay Description:Antagonist activity at human recombinant bradykinin 2 receptor expressed in CHO cells assessed as inhibition of bradykinin-induced intracellular calc...More data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
National Institute Of Neuroscienc
Curated by ChEMBL
National Institute Of Neuroscienc
Curated by ChEMBL
Affinity DataEC50: 0.0490nMAssay Description:Antagonist activity at human recombinant bradykinin 2 receptor expressed in CHO cells assessed as inhibition of bradykinin-induced intracellular calc...More data for this Ligand-Target Pair
Affinity DataEC50: 4.10nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 23nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 54nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 55nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 56nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 59nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 130nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 220nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 260nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 290nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 350nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 400nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 450nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 480nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 660nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 1.10E+3nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 1.30E+3nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+4nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair