Affinity DataEC50: 300nMAssay Description:Functional antagonism at the NMDA receptor-ion channel complex was demonstrated by the ability to inhibit the binding of thechannel-blocking agent [3...More data for this Ligand-Target Pair
Affinity DataEC50: 330nMAssay Description:Functional antagonism at the N-methyl-D-aspartate glutamate receptor 1 was demonstrated by the ability to inhibit the binding of thechannel-blocking ...More data for this Ligand-Target Pair
Affinity DataEC50: 450nMAssay Description:Activity at rat NR1/NR2D receptor expressed in Xenopus oocytes assessed as effect on glutamate-induced current by two voltage clamp electrophysiologyMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Activity at rat recombinant NR1/NR2C receptor expressed in Xenopus oocytes assessed as effect on glutamate-induced current by two voltage clamp elect...More data for this Ligand-Target Pair
Affinity DataEC50: 1.35E+3nMAssay Description:Functional antagonism at the N-methyl-D-aspartate glutamate receptor 1 was demonstrated by the ability to inhibit the binding of thechannel-blocking ...More data for this Ligand-Target Pair
Affinity DataEC50: 1.50E+3nMAssay Description:Functional antagonism at the N-methyl-D-aspartate glutamate receptor 1 was demonstrated by the ability to inhibit the binding of thechannel-blocking ...More data for this Ligand-Target Pair
Affinity DataEC50: 1.80E+3nMAssay Description:Activity at rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as effect on glutamate-induced current by two voltage clamp elect...More data for this Ligand-Target Pair
Affinity DataEC50: 2.72E+3nMAssay Description:Isolated primary cerebellum granule cells of infant rats were inoculated in 96-well plates with 1.2×105/well by using 10% FBS+25 mM KCl+2 mM Glutamin...More data for this Ligand-Target Pair
Affinity DataEC50: 2.90E+3nMAssay Description:Activity at rat recombinant NR1/NR2A receptor expressed in Xenopus oocytes assessed as effect on glutamate-induced current by two voltage clamp elect...More data for this Ligand-Target Pair
Affinity DataEC50: 2.90E+3nMAssay Description:Functional antagonism at the N-methyl-D-aspartate glutamate receptor 1 was demonstrated by the ability to inhibit the binding of thechannel-blocking ...More data for this Ligand-Target Pair
Affinity DataEC50: 3.18E+3nMAssay Description:Functional antagonism at the N-methyl-D-aspartate glutamate receptor 1 was demonstrated by the ability to inhibit the binding of thechannel-blocking ...More data for this Ligand-Target Pair
Affinity DataEC50: 3.70E+3nMAssay Description:Functional antagonism at the N-methyl-D-aspartate glutamate receptor 1 was demonstrated by the ability to inhibit the binding of thechannel-blocking ...More data for this Ligand-Target Pair
Affinity DataEC50: 4.37E+3nMAssay Description:Isolated primary cerebellum granule cells of infant rats were inoculated in 96-well plates with 1.2×105/well by using 10% FBS+25 mM KCl+2 mM Glutamin...More data for this Ligand-Target Pair
Affinity DataEC50: 4.90E+3nMAssay Description:Functional antagonism at the N-methyl-D-aspartate glutamate receptor 1 was demonstrated by the ability to inhibit the binding of thechannel-blocking ...More data for this Ligand-Target Pair
Affinity DataEC50: 5.20E+3nMAssay Description:Isolated primary cerebellum granule cells of infant rats were inoculated in 96-well plates with 1.2×105/well by using 10% FBS+25 mM KCl+2 mM Glutamin...More data for this Ligand-Target Pair
Affinity DataEC50: 5.86E+3nMAssay Description:Isolated primary cerebellum granule cells of infant rats were inoculated in 96-well plates with 1.2×105/well by using 10% FBS+25 mM KCl+2 mM Glutamin...More data for this Ligand-Target Pair
Affinity DataEC50: 6.06E+3nMAssay Description:Isolated primary cerebellum granule cells of infant rats were inoculated in 96-well plates with 1.2×105/well by using 10% FBS+25 mM KCl+2 mM Glutamin...More data for this Ligand-Target Pair
Affinity DataEC50: 7.80E+3nMAssay Description:Functional antagonism at the N-methyl-D-aspartate glutamate receptor 1 was demonstrated by the ability to inhibit the binding of thechannel-blocking ...More data for this Ligand-Target Pair
Affinity DataEC50: 8.12E+3nMAssay Description:Isolated primary cerebellum granule cells of infant rats were inoculated in 96-well plates with 1.2×105/well by using 10% FBS+25 mM KCl+2 mM Glutamin...More data for this Ligand-Target Pair
Affinity DataEC50: 8.30E+3nMAssay Description:Activity at rat NR1/NR2D receptor expressed in Xenopus oocytes assessed as effect on glutamate-induced current by two voltage clamp electrophysiologyMore data for this Ligand-Target Pair
Affinity DataEC50: 9.30E+3nMAssay Description:Isolated primary cerebellum granule cells of infant rats were inoculated in 96-well plates with 1.2×105/well by using 10% FBS+25 mM KCl+2 mM Glutamin...More data for this Ligand-Target Pair
Affinity DataEC50: 1.40E+4nMAssay Description:Activity at rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as effect on glutamate-induced current by two voltage clamp elect...More data for this Ligand-Target Pair
Affinity DataEC50: 1.54E+4nMAssay Description:Isolated primary cerebellum granule cells of infant rats were inoculated in 96-well plates with 1.2×105/well by using 10% FBS+25 mM KCl+2 mM Glutamin...More data for this Ligand-Target Pair
Affinity DataEC50: 2.20E+4nMAssay Description:Activity at rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as effect on glutamate-induced current by two voltage clamp elect...More data for this Ligand-Target Pair
Affinity DataEC50: 2.21E+4nMAssay Description:Functional antagonism at the N-methyl-D-aspartate glutamate receptor 1 was demonstrated by the ability to inhibit the binding of thechannel-blocking ...More data for this Ligand-Target Pair
Affinity DataEC50: 2.30E+4nMAssay Description:Activity at rat recombinant NR1/NR2C receptor expressed in Xenopus oocytes assessed as effect on glutamate-induced current by two voltage clamp elect...More data for this Ligand-Target Pair
Affinity DataEC50: 2.46E+4nMAssay Description:Isolated primary cerebellum granule cells of infant rats were inoculated in 96-well plates with 1.2×105/well by using 10% FBS+25 mM KCl+2 mM Glutamin...More data for this Ligand-Target Pair
Affinity DataEC50: 2.52E+4nMAssay Description:Isolated primary cerebellum granule cells of infant rats were inoculated in 96-well plates with 1.2×105/well by using 10% FBS+25 mM KCl+2 mM Glutamin...More data for this Ligand-Target Pair
Affinity DataEC50: 3.14E+4nMAssay Description:Isolated primary cerebellum granule cells of infant rats were inoculated in 96-well plates with 1.2×105/well by using 10% FBS+25 mM KCl+2 mM Glutamin...More data for this Ligand-Target Pair
Affinity DataEC50: 3.25E+4nMAssay Description:Functional antagonism at the N-methyl-D-aspartate glutamate receptor 1 was demonstrated by the ability to inhibit the binding of thechannel-blocking ...More data for this Ligand-Target Pair
Affinity DataEC50: 3.40E+4nMAssay Description:Activity at rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as effect on glutamate-induced current by two voltage clamp elect...More data for this Ligand-Target Pair
Affinity DataEC50: 3.60E+4nMAssay Description:Activity at rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as effect on glutamate-induced current by two voltage clamp elect...More data for this Ligand-Target Pair
Affinity DataEC50: 4.30E+4nMAssay Description:Activity at rat NR1/NR2D receptor expressed in Xenopus oocytes assessed as effect on glutamate-induced current by two voltage clamp electrophysiologyMore data for this Ligand-Target Pair
Affinity DataEC50: 4.70E+4nMAssay Description:Activity at rat recombinant NR1/NR2A receptor expressed in Xenopus oocytes assessed as effect on glutamate-induced current by two voltage clamp elect...More data for this Ligand-Target Pair
Affinity DataEC50: 4.80E+4nMAssay Description:Activity at rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as effect on glutamate-induced current by two voltage clamp elect...More data for this Ligand-Target Pair
Affinity DataEC50: 5.40E+4nMAssay Description:Activity at rat recombinant NR1/NR2C receptor expressed in Xenopus oocytes assessed as effect on glutamate-induced current by two voltage clamp elect...More data for this Ligand-Target Pair
Affinity DataEC50: 5.80E+4nMAssay Description:Activity at rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as effect on glutamate-induced current by two voltage clamp elect...More data for this Ligand-Target Pair
Affinity DataEC50: 6.30E+4nMAssay Description:Activity at rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as effect on glutamate-induced current by two voltage clamp elect...More data for this Ligand-Target Pair
Affinity DataEC50: 6.80E+4nMAssay Description:Activity at rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as effect on glutamate-induced current by two voltage clamp elect...More data for this Ligand-Target Pair
Affinity DataEC50: 6.90E+4nMAssay Description:Functional antagonism at the N-methyl-D-aspartate glutamate receptor 1 was demonstrated by the ability to inhibit the binding of thechannel-blocking ...More data for this Ligand-Target Pair
Affinity DataEC50: 7.50E+4nMAssay Description:Activity at rat recombinant NR1/NR2A receptor expressed in Xenopus oocytes assessed as effect on glutamate-induced current by two voltage clamp elect...More data for this Ligand-Target Pair
Affinity DataEC50: 8.20E+4nMAssay Description:Activity at rat recombinant NR1/NR2A receptor expressed in Xenopus oocytes assessed as effect on glutamate-induced current by two voltage clamp elect...More data for this Ligand-Target Pair
Affinity DataEC50: 9.10E+4nMAssay Description:Activity at rat recombinant NR1/NR2C receptor expressed in Xenopus oocytes assessed as effect on glutamate-induced current by two voltage clamp elect...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Functional antagonism at the N-methyl-D-aspartate glutamate receptor 1 was demonstrated by the ability to inhibit the binding of thechannel-blocking ...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Functional antagonism at the N-methyl-D-aspartate glutamate receptor 1 was demonstrated by the ability to inhibit the binding of thechannel-blocking ...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Functional antagonism at the N-methyl-D-aspartate glutamate receptor 1 was demonstrated by the ability to inhibit the binding of thechannel-blocking ...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Functional antagonism at the N-methyl-D-aspartate glutamate receptor 1 was demonstrated by the ability to inhibit the binding of thechannel-blocking ...More data for this Ligand-Target Pair
Affinity DataEC50: 1.05E+5nMAssay Description:Activity at rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as effect on glutamate-induced current by two voltage clamp elect...More data for this Ligand-Target Pair
Affinity DataEC50: 1.49E+5nMAssay Description:Activity at rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as effect on glutamate-induced current by two voltage clamp elect...More data for this Ligand-Target Pair
Affinity DataEC50: 1.52E+5nMAssay Description:Activity at rat NR1/NR2D receptor expressed in Xenopus oocytes assessed as effect on glutamate-induced current by two voltage clamp electrophysiologyMore data for this Ligand-Target Pair