Found 707 of ec50 data for polymerid = 50000270,50003994 
Affinity DataEC50: >0.00100nMAssay Description:Transcriptional activation of Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
Affinity DataEC50: >0.00100nMAssay Description:Transcriptional activation of Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
Affinity DataEC50: >0.00100nMAssay Description:Transcriptional activation of Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
Affinity DataEC50: 0.200nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataEC50: 0.800nMAssay Description:Activation of Nurr1 expressed in MN9D cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.900nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.900nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.40nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.5nMAssay Description:Compound was tested for functional activity in CV-1 cells transfected with an expression vector for retinoid X receptor alpha using transactivation a...More data for this Ligand-Target Pair
Affinity DataEC50: 1.5nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataEC50: 1.80nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.80nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.80nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Inhibition of Retinoic acid receptor RXR-alpha agonist activity in vitroMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Inhibition of Retinoic acid receptor RXR-alpha agonist activity in vitroMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Transcriptional ativation of Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Effective concentration required for agonistic activity in CV-1 cells expressing RXR-alphaMore data for this Ligand-Target Pair
Affinity DataEC50: 2.10nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.30nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.70nMAssay Description:Agonist activity at human RXRalpha LBD by cell based luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Effective concentration for Retinoid X receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Effective concentration for Retinoid X receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 3.30nMAssay Description:Antagonist activity against Retinoic acid receptor RXR-alpha expressed in CV-1 cell transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.40nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.40nMAssay Description:Antagonist activity against Retinoic acid receptor RXR-alpha expressed in CV-1 cell transcriptional activation assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataEC50: 3.5nMAssay Description:Activation of Nurr1 expressed in MN9D cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.80nMAssay Description:Partial agonist activity at RXRalpha (unknown origin) expressed in COS1 cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataEC50: 3.90nMAssay Description:Activation of Nurr1 expressed in MN9D cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Agonist activity for retinoic acid receptor RXR alpha in transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Ability to activate gene expression at Retinoic acid receptor RXR-alpha was evaluated in a cotransfection assay.More data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Agonist activity at human RXR-alphaMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Effective potency in transcriptional activation assay in CV-1 cells expressing retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Effective concentration for lipogenesis induced by retinoid X receptor alpha in C3H10T1/2 clone 8 fibroblast cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Effective concentration for lipogenesis induced by retinoid X receptor alpha in C3H10T1/2 clone 8 fibroblast cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Effective concentration for antagonistic activity against RXR-alpha expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Effective concentration for Retinoid X receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataEC50: 4.10nMAssay Description:Activation of Nurr1 expressed in MN9D cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Effective concentration for Retinoid X receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Effective concentration for lipogenesis induced by retinoid X receptor alpha in C3H10T1/2 clone 8 fibroblast cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Transcriptional activity was evaluated in CV-1 cells transfected with expression vector for Retinoic acid receptor RXR-alphaMore data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Transcriptional ativation of Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Transcriptional activity was evaluated in CV-1 cells transfected with expression vector for Retinoic acid receptor RXR-alphaMore data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.28nMAssay Description:Agonist activity at RXRalpha by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.30nMAssay Description:Agonist activity at RXRalpha transfected in human COS1 cells after 18 hrs by luciferase reporter gene transactivation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Ability to activate gene expression at Retinoic acid receptor RXR-alpha was evaluated in a cotransfection assay.More data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Agonist activity at human RXR-alpha expressed in U2OS cells by PathHunter assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Effective concentration against Retinoic acid receptor RXR-alphaMore data for this Ligand-Target Pair
