Compile Data Set for Download or QSAR
maximum 50k data
Found 409 of ec50 data for polymerid = 50000665,50000684,50007600,50007686,50007843,507
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50242740(CHEMBL459850 | N-(3-(7-Amino-1-methyl-2-oxo-1,2-di...)
Affinity DataEC50:  5nMAssay Description:Inhibition of Lck by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340160((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340162((S)-4-(8-amino-3-(1-but-2- ynoylpiperidin-2-yl)imi...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340167((S,E)-4-(8-amino-3-(1-(4- (dimethylamino)-N-methyl...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340079((S,E)-4-(8-amino-3-(1- cinnamoylpyrrolidin-2- yl)i...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340185((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340187((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340188((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340189((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340195((S)-4-(8-amino-3-(1-but-2- ynoylpyrrolidin-2-yl)im...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340196((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340095((S)-4-(8-amino-3-(1-but-2- ynoylpyrrolidin-2-yl)im...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme (Millipore catalog #14-442), is diluted to 0.4 U/mL in KR buffer (10 mM Tris-HCl, 10 mM MgCl2, 0.01% Tween-20, 0.05% NaN3, 1 mM DTT, 2 mM ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340160((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme (Millipore catalog #14-442), is diluted to 0.4 U/mL in KR buffer (10 mM Tris-HCl, 10 mM MgCl2, 0.01% Tween-20, 0.05% NaN3, 1 mM DTT, 2 mM ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340162((S)-4-(8-amino-3-(1-but-2- ynoylpiperidin-2-yl)imi...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme (Millipore catalog #14-442), is diluted to 0.4 U/mL in KR buffer (10 mM Tris-HCl, 10 mM MgCl2, 0.01% Tween-20, 0.05% NaN3, 1 mM DTT, 2 mM ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340167((S,E)-4-(8-amino-3-(1-(4- (dimethylamino)-N-methyl...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme (Millipore catalog #14-442), is diluted to 0.4 U/mL in KR buffer (10 mM Tris-HCl, 10 mM MgCl2, 0.01% Tween-20, 0.05% NaN3, 1 mM DTT, 2 mM ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340079((S,E)-4-(8-amino-3-(1- cinnamoylpyrrolidin-2- yl)i...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme (Millipore catalog #14-442), is diluted to 0.4 U/mL in KR buffer (10 mM Tris-HCl, 10 mM MgCl2, 0.01% Tween-20, 0.05% NaN3, 1 mM DTT, 2 mM ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340185((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme (Millipore catalog #14-442), is diluted to 0.4 U/mL in KR buffer (10 mM Tris-HCl, 10 mM MgCl2, 0.01% Tween-20, 0.05% NaN3, 1 mM DTT, 2 mM ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340187((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme (Millipore catalog #14-442), is diluted to 0.4 U/mL in KR buffer (10 mM Tris-HCl, 10 mM MgCl2, 0.01% Tween-20, 0.05% NaN3, 1 mM DTT, 2 mM ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340188((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme (Millipore catalog #14-442), is diluted to 0.4 U/mL in KR buffer (10 mM Tris-HCl, 10 mM MgCl2, 0.01% Tween-20, 0.05% NaN3, 1 mM DTT, 2 mM ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340189((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme (Millipore catalog #14-442), is diluted to 0.4 U/mL in KR buffer (10 mM Tris-HCl, 10 mM MgCl2, 0.01% Tween-20, 0.05% NaN3, 1 mM DTT, 2 mM ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340195((S)-4-(8-amino-3-(1-but-2- ynoylpyrrolidin-2-yl)im...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme (Millipore catalog #14-442), is diluted to 0.4 U/mL in KR buffer (10 mM Tris-HCl, 10 mM MgCl2, 0.01% Tween-20, 0.05% NaN3, 1 mM DTT, 2 mM ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340196((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme (Millipore catalog #14-442), is diluted to 0.4 U/mL in KR buffer (10 mM Tris-HCl, 10 mM MgCl2, 0.01% Tween-20, 0.05% NaN3, 1 mM DTT, 2 mM ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340095((S)-4-(8-amino-3-(1-but-2- ynoylpyrrolidin-2-yl)im...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340160((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340162((S)-4-(8-amino-3-(1-but-2- ynoylpiperidin-2-yl)imi...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340167((S,E)-4-(8-amino-3-(1-(4- (dimethylamino)-N-methyl...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340079((S,E)-4-(8-amino-3-(1- cinnamoylpyrrolidin-2- yl)i...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340185((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340187((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340188((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340189((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340195((S)-4-(8-amino-3-(1-but-2- ynoylpyrrolidin-2-yl)im...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340196((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340095((S)-4-(8-amino-3-(1-but-2- ynoylpyrrolidin-2-yl)im...)
Affinity DataEC50:  550nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM482158(BDBM50242742 | TAE684)
Affinity DataEC50: >1.00E+3nMAssay Description:Inhibition of Lck by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340118(US10239883, Example 1 | US10934296, Example 1 | US...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340080(US9758524, Example 2)
Affinity DataEC50: >1.00E+3nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340119(US10239883, Example 3 | US10934296, Example 3 | US...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340081(US10239883, Example 4 | US10934296, Example 4 | US...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340082(US10239883, Example 5 | US10934296, Example 5 | US...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50175583(ACP-196 | Acalabrutinib | US10239883, Example 6 | ...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340083(US10239883, Example 7 | US10934296, Example 7 | US...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340121(US10239883, Example 8 | US10934296, Example 8 | US...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340122(US10239883, Example 9 | US10934296, Example 9 | US...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340123(US10239883, Example 10 | US10934296, Example 10 | ...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340084(US10239883, Example 11 | US10934296, Example 11 | ...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340124(US10239883, Example 12 | US10934296, Example 12 | ...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340125(US10934296, Example 13 | US9758524, Example 13)
Affinity DataEC50: >1.00E+3nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340126(US10239883, Example 14 | US10934296, Example 14 | ...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM340127(US10239883, Example 15 | US10934296, Example 15 | ...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lck enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lck enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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