Affinity DataEC50: 0.0680nMAssay Description:Agonist activity at human OX1R expressed in CHO-K1 cells by FLIPR calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.130nMAssay Description:Agonist activity at OX1 receptor (unknown origin) expressed in RD-HGA16 cells assessed as calcium mobilization by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.220nMAssay Description:Agonist activity at human OX1 receptor overexpressed in CHO-RD-HGA16 cells assessed as calcium mobilization after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.410nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.520nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.610nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.770nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.820nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.830nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.850nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.890nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 1.10nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 1.30nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 1.40nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 1.40nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 1.40nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 1.5nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 1.60nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 1.60nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 1.70nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 2.30nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 2.30nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 2.40nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 2.60nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 2.70nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 2.70nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 3.10nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 3.20nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 3.40nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 3.80nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 4.80nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 5.70nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 5.80nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 7nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 7.30nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 7.5nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 7.90nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 8.10nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 8.30nMAssay Description:Agonist activity at human OX1 receptor overexpressed in CHO-RD-HGA16 cells assessed as calcium mobilization after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 9.10nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 9.80nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:Agonist activity at OX1R (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 22nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 22nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
Affinity DataEC50: 24nMAssay Description:Agonist activity at human OX1R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair